Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50009426
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083523((1-Benzyl-1H-quinolin-4-ylidene)-pentyl-amine | CH...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083514(4-[(E)-2-(3,4-Bis-benzyloxy-phenyl)-vinyl]-4'-chlo...)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083518(4'-Chloro-4-((E)-4-phenyl-but-1-enyl)-biphenyl-2-c...)
Affinity DataIC50:  3.20E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083522(4'-Chloro-4-[(E)-2-(4-chloro-3-fluoro-phenyl)-viny...)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083515(2-({4'-chloro-4-[(E)-2-(4-fluorophenyl)vinyl]-1,1'...)
Affinity DataIC50:  3.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083513(4'-Chloro-4-((E)-4-phenyl-but-1-enyl)-biphenyl-2-c...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083511(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083516(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  5.80E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083519(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  6.10E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083517(4'-Chloro-4-[(E)-2-(2-fluoro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  8.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083512(4'-Chloro-4-[(E)-2-(4-fluoro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  9.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083520(4-[(E)-2-(4-Benzyloxy-phenyl)-vinyl]-4'-chloro-bip...)
Affinity DataIC50:  9.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50083521(4'-Chloro-4-[(E)-2-(3-chloro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  1.01E+4nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed