Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50035031
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.0620nMAssay Description:Ability to inhibit binding of SNC80 to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.220nMAssay Description:Ability to displace [3H]U-69593 from kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  3.20nMAssay Description:Ability to displace [3H]DADL from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  6.60nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  8.85nMAssay Description:Ability to inhibit binding of U-69,593 to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  8.90nMAssay Description:Ability to displace [3H]DADL from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  9nMAssay Description:Ability to inhibit binding of SNC80 to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  27nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366621(CHEMBL1743886)
Affinity DataKi:  99nMAssay Description:Ability to displace [3H]DADL from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50083727(16-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-dia...)
Affinity DataKi:  103nMAssay Description:Ability to displace [3H]DADL from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50083727(16-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-dia...)
Affinity DataKi:  396nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  411nMAssay Description:Ability to inhibit binding of [3H]DAMGO to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50083727(16-benzyloxy-22-cyclopropylmethyl-14-oxa-11,22-dia...)
Affinity DataKi:  728nMAssay Description:Ability to displace [3H]U-69593 from kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366622(CHEMBL1202098)
Affinity DataKi:  1.04E+3nMAssay Description:Ability to displace [3H]DADL from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  1.76E+3nMAssay Description:Ability to inhibit binding of U-69,593 to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  2.51E+3nMAssay Description:Ability to inhibit binding of [3H]DAMGO to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366623(CHEMBL1744389)
Affinity DataKi:  3.91E+3nMAssay Description:Ability to displace [3H]U-69593 from kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366621(CHEMBL1743886)
Affinity DataKi: >5.32E+3nMAssay Description:Ability to displace [3H]U-69593 from kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366622(CHEMBL1202098)
Affinity DataKi: >6.25E+3nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366621(CHEMBL1743886)
Affinity DataKi: >6.25E+3nMAssay Description:Ability to displace [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366622(CHEMBL1202098)
Affinity DataKi: >7.04E+3nMAssay Description:Ability to displace [3H]U-69593 from kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed