Compile Data Set for Download or QSAR
maximum 50k data
Found 73 Enz. Inhib. hit(s) with all data for entry = 50009454
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083743(1N-[1-amino(imino)methyl-6-hydroxy-(5S)-tetrahydro...)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083747(CHEMBL325869 | Cinnoline-4-carboxylic acid ((R)-3-...)
Affinity DataIC50:  4.20nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083756(CHEMBL117092 | Isoquinoline-1-carboxylic acid ((R)...)
Affinity DataIC50:  4.90nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083754(CHEMBL420688 | Pyrazine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083747(CHEMBL325869 | Cinnoline-4-carboxylic acid ((R)-3-...)
Affinity DataIC50:  5.60nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083744(CHEMBL331807 | N-((R)-3-{[((S)-1-Carbamimidoyl-2-h...)
Affinity DataIC50:  6.10nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083750(CHEMBL115902 | Quinoline-3-carboxylic acid ((R)-3-...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083751(CHEMBL420322 | Pyrazine-2-carboxylic acid ((R)-4-{...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083742(CHEMBL324485 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083749(CHEMBL323642 | Pyridine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083744(CHEMBL331807 | N-((R)-3-{[((S)-1-Carbamimidoyl-2-h...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083753(CHEMBL116245 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083740(((R)-3-[(5-Bromo-pyridine-3-carbonyl)-amino]-1-{[(...)
Affinity DataIC50: >31nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083739(CHEMBL115707 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083746(CHEMBL117716 | Quinoline-2-carboxylic acid ((R)-3-...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083746(CHEMBL117716 | Quinoline-2-carboxylic acid ((R)-3-...)
Affinity DataIC50:  59nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083743(1N-[1-amino(imino)methyl-6-hydroxy-(5S)-tetrahydro...)
Affinity DataIC50:  75nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083741(CHEMBL419222 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  75nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083752(CHEMBL117678 | N-((R)-3-{[((S)-1-Carbamimidoyl-2-h...)
Affinity DataIC50:  79nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083756(CHEMBL117092 | Isoquinoline-1-carboxylic acid ((R)...)
Affinity DataIC50:  98nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083753(CHEMBL116245 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  106nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083739(CHEMBL115707 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  106nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083750(CHEMBL115902 | Quinoline-3-carboxylic acid ((R)-3-...)
Affinity DataIC50:  111nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083748(CHEMBL117721 | Pyrazine-2-carboxylic acid ((R)-2-{...)
Affinity DataIC50:  152nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083754(CHEMBL420688 | Pyrazine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  166nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083742(CHEMBL324485 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  169nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083749(CHEMBL323642 | Pyridine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  223nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083750(CHEMBL115902 | Quinoline-3-carboxylic acid ((R)-3-...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083748(CHEMBL117721 | Pyrazine-2-carboxylic acid ((R)-2-{...)
Affinity DataIC50:  311nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083738(CHEMBL115378 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  313nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083740(((R)-3-[(5-Bromo-pyridine-3-carbonyl)-amino]-1-{[(...)
Affinity DataIC50:  313nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083751(CHEMBL420322 | Pyrazine-2-carboxylic acid ((R)-4-{...)
Affinity DataIC50:  324nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083741(CHEMBL419222 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  346nMAssay Description:In vitro inhibition of human Factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083744(CHEMBL331807 | N-((R)-3-{[((S)-1-Carbamimidoyl-2-h...)
Affinity DataIC50:  367nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083754(CHEMBL420688 | Pyrazine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  521nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083750(CHEMBL115902 | Quinoline-3-carboxylic acid ((R)-3-...)
Affinity DataIC50:  537nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083752(CHEMBL117678 | N-((R)-3-{[((S)-1-Carbamimidoyl-2-h...)
Affinity DataIC50:  561nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083751(CHEMBL420322 | Pyrazine-2-carboxylic acid ((R)-4-{...)
Affinity DataIC50:  673nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083747(CHEMBL325869 | Cinnoline-4-carboxylic acid ((R)-3-...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083756(CHEMBL117092 | Isoquinoline-1-carboxylic acid ((R)...)
Affinity DataIC50:  730nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083745(5-Bromo-N-((R)-3-{[((S)-1-carbamimidoyl-2-hydroxy-...)
Affinity DataIC50:  1.06E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083742(CHEMBL324485 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  1.14E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083749(CHEMBL323642 | Pyridine-2-carboxylic acid ((R)-3-{...)
Affinity DataIC50:  1.14E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083746(CHEMBL117716 | Quinoline-2-carboxylic acid ((R)-3-...)
Affinity DataIC50:  1.27E+3nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083746(CHEMBL117716 | Quinoline-2-carboxylic acid ((R)-3-...)
Affinity DataIC50:  1.44E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083748(CHEMBL117721 | Pyrazine-2-carboxylic acid ((R)-2-{...)
Affinity DataIC50:  1.48E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083747(CHEMBL325869 | Cinnoline-4-carboxylic acid ((R)-3-...)
Affinity DataIC50:  1.77E+3nMAssay Description:In vitro inhibition of human Thrombin (FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50083753(CHEMBL116245 | {(R)-1-{[((S)-1-Carbamimidoyl-2-hyd...)
Affinity DataIC50:  2.03E+3nMAssay Description:In vitro inhibition of human thrombolytic protease Plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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