Compile Data Set for Download or QSAR
maximum 50k data
Found 135 Enz. Inhib. hit(s) with all data for entry = 50009495
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17284(2-{[2-(5-carbamimidoyl-2-hydroxyphenoxy)-3,5-diflu...)
Affinity DataKi:  0.110nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17277((Z,Z)BABCH | 4-{[(1Z,3Z)-3-[(4-carbamimidoylphenyl...)
Affinity DataKi:  0.660nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084175(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(Z)-ylide...)
Affinity DataKi:  2.5nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084186(2,9-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  2.80nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084174(2,8-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  4.60nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084192(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(Z)-ylide...)
Affinity DataKi:  4.80nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084163(2,6-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  5.20nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066616((Z,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  5.60nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084170(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(Z)-ylide...)
Affinity DataKi:  6.90nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084164(2-[1-[4-amino(imino)methylphenyl]-(Z)-methylidene]...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084160(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  15nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084177(2-[1-[4-amino(imino)methylphenyl]-(Z)-methylidene]...)
Affinity DataKi:  18nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084176(2,6-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  18nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084175(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(Z)-ylide...)
Affinity DataKi:  20nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  29nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084164(2-[1-[4-amino(imino)methylphenyl]-(Z)-methylidene]...)
Affinity DataKi:  30nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084191(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  30nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17277((Z,Z)BABCH | 4-{[(1Z,3Z)-3-[(4-carbamimidoylphenyl...)
Affinity DataKi:  33nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataKi:  40nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066616((Z,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  44nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084180(4-[3-[1-(4-Carbamimidoyl-phenyl)-meth-(Z)-ylidene]...)
Affinity DataKi:  50nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084160(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  52nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084193(2,6-di[1-[4-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  56nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084183(3-[1-(4-Carbamimidoyl-phenyl)-meth-(E)-ylidene]-5-...)
Affinity DataKi:  61nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084178(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(E)-ylide...)
Affinity DataKi:  72nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084177(2-[1-[4-amino(imino)methylphenyl]-(Z)-methylidene]...)
Affinity DataKi:  90nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084192(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(Z)-ylide...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084174(2,8-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084163(2,6-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084188(2,10-di[1-[4-amino(imino)methylphenyl]-(Z)-methyli...)
Affinity DataKi:  110nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084180(4-[3-[1-(4-Carbamimidoyl-phenyl)-meth-(Z)-ylidene]...)
Affinity DataKi:  110nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084160(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084173(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084161(3,5-Bis-[1-(4-carbamimidoyl-phenyl)-meth-(E)-ylide...)
Affinity DataKi:  125nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  130nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084191(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  130nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066613((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  140nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084179(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  150nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084165(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  155nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084189(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  160nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084162(2,6-di[1-[4-amino(imino)methylphenyl]-(E)-methylid...)
Affinity DataKi:  170nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084186(2,9-di[1-[4-amino(imino)methylphenyl]-(Z)-methylid...)
Affinity DataKi:  190nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084191(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  200nMAssay Description:In vitro inhibition of human thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066613((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  200nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066615((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  200nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084158(3-[1-(4-Carbamimidoyl-phenyl)-meth-(E)-ylidene]-5-...)
Affinity DataKi:  224nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084183(3-[1-(4-Carbamimidoyl-phenyl)-meth-(E)-ylidene]-5-...)
Affinity DataKi:  225nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084187(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  230nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50084173(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  260nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50066614((E,E)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  280nMAssay Description:In vitro inhibition of bovine trypsin(Trp).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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