Compile Data Set for Download or QSAR
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Found 36 Enz. Inhib. hit(s) with all data for entry = 50009866
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088706(CHEMBL12062 | N-{3-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088702(CHEMBL275469 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088704(1-{(E)-5-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-...)
Affinity DataKi:  18nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088703(CHEMBL12603 | N-{2-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  18nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088707(1-({2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-eth...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088700(1-{4-Hydroxy-5-[4-(2-isopropoxy-phenyl)-piperazin-...)
Affinity DataKi:  28nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088705((2-Oxo-piperidin-1-yl)-acetic acid 2-[4-(2-isoprop...)
Affinity DataKi:  38nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088698(CHEMBL268030 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  53nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088706(CHEMBL12062 | N-{3-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  80nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088697(CHEMBL418531 | N-{2-[4-(4-Fluoro-2-isopropoxy-phen...)
Affinity DataKi:  83nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088708(CHEMBL12501 | N-{3-[4-(2-Methoxy-phenyl)-piperazin...)
Affinity DataKi:  98nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088705((2-Oxo-piperidin-1-yl)-acetic acid 2-[4-(2-isoprop...)
Affinity DataKi:  108nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088701(CHEMBL12364 | N-(2-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
Affinity DataKi:  129nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088700(1-{4-Hydroxy-5-[4-(2-isopropoxy-phenyl)-piperazin-...)
Affinity DataKi:  253nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088707(1-({2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-eth...)
Affinity DataKi:  260nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088702(CHEMBL275469 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  372nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088699(1-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-5-(2-ox...)
Affinity DataKi:  417nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088703(CHEMBL12603 | N-{2-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  505nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088704(1-{(E)-5-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-...)
Affinity DataKi:  602nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088698(CHEMBL268030 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  650nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088705((2-Oxo-piperidin-1-yl)-acetic acid 2-[4-(2-isoprop...)
Affinity DataKi:  2.24E+3nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088703(CHEMBL12603 | N-{2-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  3.54E+3nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088697(CHEMBL418531 | N-{2-[4-(4-Fluoro-2-isopropoxy-phen...)
Affinity DataKi:  4.50E+3nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088704(1-{(E)-5-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-...)
Affinity DataKi:  5.32E+3nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088701(CHEMBL12364 | N-(2-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
Affinity DataKi:  5.35E+3nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088699(1-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-5-(2-ox...)
Affinity DataKi:  6.04E+3nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088700(1-{4-Hydroxy-5-[4-(2-isopropoxy-phenyl)-piperazin-...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088699(1-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-5-(2-ox...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088701(CHEMBL12364 | N-(2-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088697(CHEMBL418531 | N-{2-[4-(4-Fluoro-2-isopropoxy-phen...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088706(CHEMBL12062 | N-{3-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088698(CHEMBL268030 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088708(CHEMBL12501 | N-{3-[4-(2-Methoxy-phenyl)-piperazin...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088708(CHEMBL12501 | N-{3-[4-(2-Methoxy-phenyl)-piperazin...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088707(1-({2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-eth...)
Affinity DataKi:  2.63E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50088702(CHEMBL275469 | N-{2-[4-(2-Isopropoxy-phenyl)-piper...)
Affinity DataKi:  4.61E+4nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed