Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50009917
TargetNeutrophil elastase(Homo sapiens (Human))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(CHEMBL266704 | Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp...)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition constant of the compound was tested against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(CHEMBL216418 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser...)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition constant of the compound was tested against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(CHEMBL216418 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser...)
Affinity DataKi:  1.00E+5nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(CHEMBL216418 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser...)
Affinity DataKi:  1.60E+5nMAssay Description:Competitive inhibition constant of the compound was tested against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(CHEMBL266704 | Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp...)
Affinity DataKi:  1.90E+5nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(CHEMBL414810 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser)
Affinity DataKi:  1.90E+5nMAssay Description:Competitive inhibition constant of the compound was tested against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(CHEMBL266704 | Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp...)
Affinity DataKi:  2.40E+5nMAssay Description:Competitive inhibition constant of the compound was tested against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089096(CHEMBL278549 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met | e...)
Affinity DataKi:  2.70E+5nMAssay Description:Competitive inhibition constant of the compound was tested against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089097(CHEMBL21028 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Lys)
Affinity DataKi:  5.40E+5nMAssay Description:Competitive inhibition constant of the compound was tested against trypsin using the reporter substrate Ac-R-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089099((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-methylsulfanyl-...)
Affinity DataKi:  1.10E+6nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089096(CHEMBL278549 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met | e...)
Affinity DataKi:  2.30E+6nMAssay Description:Competitive inhibition constant of the compound was tested against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(CHEMBL414810 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser)
Affinity DataKi:  3.10E+6nMAssay Description:Competitive inhibition constant of the compound was tested against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(CHEMBL414810 | Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser)
Affinity DataKi:  5.80E+6nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed