Compile Data Set for Download or QSAR
maximum 50k data
Found 87 Enz. Inhib. hit(s) with all data for entry = 50010046
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090310(CHEMBL44294 | N-{3-[4-(2-Chloro-phenyl)-4-cyano-pi...)
Affinity DataKi:  0.990nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090306(2,2-Di-p-tolyl-N-[3-(4-o-tolyl-piperazin-1-yl)-pro...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090307(CHEMBL298058 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090305(CHEMBL41994 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1-...)
Affinity DataKi:  2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090305(CHEMBL41994 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1-...)
Affinity DataKi:  2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090305(CHEMBL41994 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1-...)
Affinity DataKi:  2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090309(CHEMBL42514 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1-...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50068819(5-[3-(4-Methoxycarbonyl-4-phenyl-piperidin-1-yl)-p...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090304(1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090316(2-(4-Chloro-phenyl)-N-[3-(4-cyano-4-o-tolyl-piperi...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090306(2,2-Di-p-tolyl-N-[3-(4-o-tolyl-piperazin-1-yl)-pro...)
Affinity DataKi:  6.60nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090322(CHEMBL44124 | N-[3-(4-Cyano-4-phenyl-piperidin-1-y...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090318(CHEMBL297667 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090303(CHEMBL42220 | N-{3-[4-Cyano-4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  7.5nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090325(CHEMBL295304 | N-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataKi:  8.80nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090311(CHEMBL435576 | N-[3-(4-Phenyl-piperazin-1-yl)-prop...)
Affinity DataKi:  12nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090300(CHEMBL42763 | N-{3-[4-Cyano-4-(2-trifluoromethyl-p...)
Affinity DataKi:  22nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090311(CHEMBL435576 | N-[3-(4-Phenyl-piperazin-1-yl)-prop...)
Affinity DataKi:  23nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090324(CHEMBL417350 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1...)
Affinity DataKi:  24nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090313(CHEMBL432302 | N-[3-(4'-Cyano-3',4',5',6'-tetrahyd...)
Affinity DataKi:  25nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090323(CHEMBL289916 | N-[3-(3',4',5',6'-Tetrahydro-2'H-[2...)
Affinity DataKi:  27nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090312(CHEMBL296965 | N-[3-(4-Cyano-4-phenyl-piperidin-1-...)
Affinity DataKi:  28nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090325(CHEMBL295304 | N-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataKi:  34nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090306(2,2-Di-p-tolyl-N-[3-(4-o-tolyl-piperazin-1-yl)-pro...)
Affinity DataKi:  36nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090301(1-{3-[2-(4-Nitro-phenyl)-propionylamino]-propyl}-4...)
Affinity DataKi:  47nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090320(CHEMBL416073 | N-[3-(4-Cyano-4-phenyl-piperidin-1-...)
Affinity DataKi:  50nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090302(CHEMBL40303 | N-[3-(4-Cyano-4-phenyl-piperidin-1-y...)
Affinity DataKi:  61nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090321(CHEMBL42361 | N-[3-(4-Cyano-4-phenyl-piperidin-1-y...)
Affinity DataKi:  72nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090315(4-Phenyl-1-[3-(2-p-tolyl-acetylamino)-propyl]-pipe...)
Affinity DataKi:  74nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090308(1-{3-[2-(4-Nitro-phenyl)-acetylamino]-propyl}-4-ph...)
Affinity DataKi:  75nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090311(CHEMBL435576 | N-[3-(4-Phenyl-piperazin-1-yl)-prop...)
Affinity DataKi:  128nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090325(CHEMBL295304 | N-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataKi:  230nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090319(1-{3-[3-(4-Nitro-phenyl)-propionylamino]-propyl}-4...)
Affinity DataKi:  240nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090310(CHEMBL44294 | N-{3-[4-(2-Chloro-phenyl)-4-cyano-pi...)
Affinity DataKi:  280nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090307(CHEMBL298058 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1...)
Affinity DataKi:  360nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090317(1-{2-[3-(4-Nitro-phenyl)-propionylamino]-ethyl}-4-...)
Affinity DataKi:  380nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090304(1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl...)
Affinity DataKi:  450nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090303(CHEMBL42220 | N-{3-[4-Cyano-4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  570nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090314(1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl...)
Affinity DataKi:  570nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090314(1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl...)
Affinity DataKi:  570nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090310(CHEMBL44294 | N-{3-[4-(2-Chloro-phenyl)-4-cyano-pi...)
Affinity DataKi:  600nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090318(CHEMBL297667 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1...)
Affinity DataKi:  650nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090323(CHEMBL289916 | N-[3-(3',4',5',6'-Tetrahydro-2'H-[2...)
Affinity DataKi:  670nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090309(CHEMBL42514 | N-[3-(4-Cyano-4-o-tolyl-piperidin-1-...)
Affinity DataKi:  680nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50068819(5-[3-(4-Methoxycarbonyl-4-phenyl-piperidin-1-yl)-p...)
Affinity DataKi:  700nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090303(CHEMBL42220 | N-{3-[4-Cyano-4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  710nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090312(CHEMBL296965 | N-[3-(4-Cyano-4-phenyl-piperidin-1-...)
Affinity DataKi:  840nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090316(2-(4-Chloro-phenyl)-N-[3-(4-cyano-4-o-tolyl-piperi...)
Affinity DataKi:  870nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090319(1-{3-[3-(4-Nitro-phenyl)-propionylamino]-propyl}-4...)
Affinity DataKi:  910nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50090304(1-[3-(2,2-Di-p-tolyl-acetylamino)-propyl]-4-phenyl...)
Affinity DataKi:  960nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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