Affinity DataKi: 0.200nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:In vivo inhibitory effect against Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:In vitro antagonism at Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 288nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 313nMAssay Description:In vivo inhibitory effect of the compound against Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 366nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 425nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 531nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 588nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 616nMAssay Description:Selectivity screen against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 682nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 805nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 842nMAssay Description:In vitro antagonism at Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:In vitro antagonism at Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 955nMAssay Description:In vivo inhibitory effect of the compound against alpha-2b Adrenergic receptorMore data for this Ligand-Target Pair