Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50010073
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090644(CHEMBL48837 | {(S)-1-[(S)-1-(4-Butoxy-benzyl)-2,3-...)
Affinity DataKi:  0.600nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090645((S)-2-Benzyl-N-[(S)-4-guanidino-1-(2-oxo-acetyl)-b...)
Affinity DataKi:  40nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090645((S)-2-Benzyl-N-[(S)-4-guanidino-1-(2-oxo-acetyl)-b...)
Affinity DataKi:  90nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090644(CHEMBL48837 | {(S)-1-[(S)-1-(4-Butoxy-benzyl)-2,3-...)
Affinity DataKi:  214nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090646((S)-2-Acetylamino-5-guanidino-pentanoic acid [(S)-...)
Affinity DataKi:  640nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090643((S)-2-Acetylamino-4-methyl-pentanoic acid {(S)-1-[...)
Affinity DataKi:  970nMAssay Description:Ability to block cathepsin L-catalyzed hydrolysis of the fluorogenic substrate Z-Phe-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Bos taurus (bovine))
Queen'S University Belfast

Curated by ChEMBL
LigandPNGBDBM50090643((S)-2-Acetylamino-4-methyl-pentanoic acid {(S)-1-[...)
Affinity DataKi:  1.25E+3nMAssay Description:Ability to block cathepsin B-catalyzed hydrolysis of the fluorogenic substrate Z-Arg-Arg-NHMecMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed