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Found 13 Enz. Inhib. hit(s) with all data for entry = 50010115
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory activity against Opioid receptor delta 1 in rat brain membranes using [3H]-DADLE as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091224(4-[(4-But-2-enyl-2,5-dimethyl-piperazin-1-yl)-(3-m...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091221(4-[(4-Butyl-2,5-dimethyl-piperazin-1-yl)-(3-methox...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091223(4-[(4-Cyclopropylmethyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091226(CHEMBL323733 | N,N-Diethyl-4-[(3-methoxy-phenyl)-(...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091225(4-[(2,5-Dimethyl-4-pentyl-piperazin-1-yl)-(3-metho...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091217(4-[(2,5-Dimethyl-piperazin-1-yl)-(3-methoxy-phenyl...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091219(4-[[2,5-Dimethyl-4-(2-methyl-allyl)-piperazin-1-yl...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091222(CHEMBL111389 | N,N-Diethyl-4-[(4-ethyl-2,5-dimethy...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091218(4-[(4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(3-metho...)
Affinity DataKi:  6.20nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091216(CHEMBL321927 | N,N-Diethyl-4-[(4-hexyl-2,5-dimethy...)
Affinity DataKi:  10.4nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091220(4-[[2,5-Dimethyl-4-(3-phenyl-propyl)-piperazin-1-y...)
Affinity DataKi:  16.7nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50091215(4-[(2,5-Dimethyl-4-phenethyl-piperazin-1-yl)-(3-me...)
Affinity DataKi:  30.6nMAssay Description:Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed