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Found 13 Enz. Inhib. hit(s) with all data for entry = 961
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  100nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7586((2E)-3-[3-(benzyloxy)phenyl]prop-2-enal | Cinnamal...)
Affinity DataIC50:  7.50E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7570((2E)-3-[2-(benzyloxy)phenyl]prop-2-enal | Cinnamal...)
Affinity DataIC50:  1.10E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7587((2E)-3-{3-[(2-methylphenyl)methoxy]phenyl}prop-2-e...)
Affinity DataIC50:  1.50E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7571((2E)-3-{2-[(2-methylphenyl)methoxy]phenyl}prop-2-e...)
Affinity DataIC50:  1.80E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7569((2E)-3-(3-hydroxyphenyl)prop-2-enal | Cinnamaldehy...)
Affinity DataIC50:  3.00E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7568((2E)-3-(2-hydroxyphenyl)prop-2-enal | Cinnamaldehy...)
Affinity DataIC50:  3.50E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7569((2E)-3-(3-hydroxyphenyl)prop-2-enal | Cinnamaldehy...)
Affinity DataIC50:  4.50E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 100 uM ATP/ [gamma-33P] ATP. 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7586((2E)-3-[3-(benzyloxy)phenyl]prop-2-enal | Cinnamal...)
Affinity DataIC50:  5.00E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7570((2E)-3-[2-(benzyloxy)phenyl]prop-2-enal | Cinnamal...)
Affinity DataIC50:  5.00E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7587((2E)-3-{3-[(2-methylphenyl)methoxy]phenyl}prop-2-e...)
Affinity DataIC50:  6.00E+4nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7568((2E)-3-(2-hydroxyphenyl)prop-2-enal | Cinnamaldehy...)
Affinity DataIC50:  1.30E+5nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Korea Research Institute Of Bioscience And Biotechnology

LigandPNGBDBM7571((2E)-3-{2-[(2-methylphenyl)methoxy]phenyl}prop-2-e...)
Affinity DataIC50:  2.00E+5nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed