Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 50010386
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094166(CHEMBL139167 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  0.75nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094131(CHEMBL138463 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094178(CHEMBL342662 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094137(CHEMBL138890 | N-[2-Benzo[1,3]dioxol-4-yl-2-(4-cyc...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094182(CHEMBL137609 | N-[2-Benzo[1,3]dioxol-4-yl-2-(4-iso...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094156(CHEMBL342607 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094171(CHEMBL140124 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094181(CHEMBL140299 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094123(CHEMBL136764 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094154(CHEMBL139015 | N-[2-Benzo[1,3]dioxol-4-yl-2-(4-cyc...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094165(CHEMBL136305 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094185(CHEMBL138825 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094168(CHEMBL137887 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094159(CHEMBL139286 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094160(CHEMBL139226 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094175(CHEMBL137580 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094144(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-cyclohe...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094141(CHEMBL136323 | N-(2-[1,4']Bipiperidinyl-1'-yl-2-ph...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094119(CHEMBL137255 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094140(CHEMBL433683 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094143(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-cyclohe...)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094157(CHEMBL136559 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094151(CHEMBL139967 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094158(CHEMBL139854 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094139(CHEMBL138764 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094134(CHEMBL344646 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094120(1-{2-[[1,4']Bipiperidinyl-1'-yl-(2-methoxy-phenyl)...)
Affinity DataIC50:  4.30nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094128(CHEMBL336261 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094149(CHEMBL139176 | N-(2-Benzo[1,3]dioxol-5-yl-2-[1,4']...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094130(CHEMBL139569 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094117(CHEMBL140023 | N-[2-{4-[Bis-(2-hydroxy-ethyl)-amin...)
Affinity DataIC50:  5.20nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094127(CHEMBL136832 | N-(2-[1,4']Bipiperidinyl-1'-yl-2-ph...)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094121(CHEMBL344378 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094179(CHEMBL139903 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  6.40nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094153(CHEMBL138853 | N-[2-Benzo[1,3]dioxol-4-yl-2-(4-iso...)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094142(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-cyclohe...)
Affinity DataIC50:  7nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094169(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(4-indan-2...)
Affinity DataIC50:  7.20nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094132(CHEMBL139190 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  7.60nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094146(CHEMBL139189 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  8.90nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094124(CHEMBL140134 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094162(CHEMBL336715 | N-[2-(3,5-Bis-trifluoromethyl-pheny...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094167(CHEMBL138715 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(2...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094122(CHEMBL344434 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094163(CHEMBL138770 | {2-[[1,4']Bipiperidinyl-1'-yl-(2-me...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094126(CHEMBL138269 | N-(2-[1,4']Bipiperidinyl-1'-yl-2-na...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094155((2-[1,4']Bipiperidinyl-1'-yl-2-phenyl-ethyl)-[2-(3...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094184(2-(3,5-Bis-trifluoromethyl-phenyl)-N-[2-(3,4-dichl...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094176(CHEMBL135028 | N-[2-(4-Cyclohexyl-piperazin-1-yl)-...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094150(CHEMBL139057 | N-(2-Benzo[1,3]dioxol-4-yl-2-[1,4']...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Biographics Laboratory 3R

Curated by ChEMBL
LigandPNGBDBM50094129(CHEMBL136544 | N-[2-[1,4']Bipiperidinyl-1'-yl-2-(3...)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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