Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 5289
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.143nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.151nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85732(Tmt-D-Arg-Phe-Lys-NH2)
Affinity DataKi:  0.192nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  0.222nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85733(H-Dmt-D-Arg-Phe-A2bu-NH2)
Affinity DataKi:  0.803nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85737(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  1.76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  2.06nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  2.53nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  9.43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  11.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  22.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  26.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  32.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85732(Tmt-D-Arg-Phe-Lys-NH2)
Affinity DataKi:  46.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85733(H-Dmt-D-Arg-Phe-A2bu-NH2)
Affinity DataKi:  47.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  193nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85732(Tmt-D-Arg-Phe-Lys-NH2)
Affinity DataKi:  543nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  1.24E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  1.84E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  2.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  2.32E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  3.94E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85737(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  4.23E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  4.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85733(H-Dmt-D-Arg-Phe-A2bu-NH2)
Affinity DataKi:  6.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi:  9.22E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM85734(H-Hmt-D-Arg-Phe-Lys-NH2 I | H-Hmt-D-Arg-Phe-Lys-NH...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed