Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50035162
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50450369(SIALYL LEWIS X | Sialyl LeX | Sialyl lewis-x | sLe...)
Affinity DataIC50:  3.00E+5nMAssay Description:In vitro inhibitory activity against binding of Selectin E to human recombinant AGP (alpha-1 acid glycoprotein) containing sLex derivativeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096284(2-{2-[6-(4-Benzyl-4-hydroxy-piperidin-1-ylmethyl)-...)
Affinity DataIC50:  1.60E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096291(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  3.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096293(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  6.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096287(5-({6-[(1,3-Dicarboxy-propylcarbamoyl)-methyl]-3,4...)
Affinity DataIC50:  6.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096290(2-(2-{6-[(1-Carbamoyl-2-phenyl-ethylamino)-methyl]...)
Affinity DataIC50:  6.70E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096292(6-Amino-2-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tet...)
Affinity DataIC50:  7.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096289(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  7.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096286(2-[2-(3,4,5-Trihydroxy-6-{[methyl-(3-methyl-cycloh...)
Affinity DataIC50:  8.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096294(4-Carbamoyl-2-[2-(3,4,5-trihydroxy-6-hydroxymethyl...)
Affinity DataIC50: >1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096285(3-{4-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahyd...)
Affinity DataIC50:  1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096288(4-{4-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahyd...)
Affinity DataIC50: >1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed