Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50010682
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of gelatinase A (Matrix metalloproteinase-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50:  20nMAssay Description:Inhibition of gelatinase A (Matrix metalloproteinase-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloproteinase-13)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50:  38nMAssay Description:Inhibition of gelatinase A (Matrix metalloproteinase-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50:  131nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloproteinase-13)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50:  176nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloproteinase-13)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  251nMAssay Description:Inhibition of gelatinase A (Matrix metalloproteinase-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  338nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloproteinase-13)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of Stomelysin (Matrix metalloproteinase-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of Stomelysin (Matrix metalloproteinase-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of Stomelysin (Matrix metalloproteinase-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50:  6.15E+3nMAssay Description:Inhibition of Stomelysin (Matrix metalloproteinase-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed