Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50010814
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099016(CHEMBL275964 | Cyclohexanecarboxylic acid {(S)-1-b...)
Affinity DataKi:  0.800nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099015(CHEMBL10796 | Cyclohexanecarboxylic acid {(R)-1-be...)
Affinity DataKi:  1.5nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099014(CHEMBL10793 | Cyclohexanecarboxylic acid {(R)-1-be...)
Affinity DataKi:  4.5nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099013(CHEMBL10603 | N-{(R)-1-Benzyl-2-[4-(4-methoxy-[1,2...)
Affinity DataKi:  9.90nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099012(CHEMBL10764 | N-{(S)-1-Benzyl-2-[4-(4-chloro-[1,2,...)
Affinity DataKi:  425nMAssay Description:Ability to displace [3H]-8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50:  489nMAssay Description:Percent inhibition of the compound towards dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50:  1.10E+3nMAssay Description:Percent inhibition of the compound towards dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50:  3.52E+3nMAssay Description:Percent inhibition of the compound towards dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed