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Found 24 Enz. Inhib. hit(s) with all data for entry = 50036959
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102880(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102880(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  1.09E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102880(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  1.28E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102880(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102880(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50263769((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...)
Affinity DataKi:  2.98E+4nMAssay Description:Inhibitory activity against liver Glycogen Phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50240802(1-N-ACETYL-BETA-D-GLUCOSAMINE | CHEMBL335315 | N-(...)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50240802(1-N-ACETYL-BETA-D-GLUCOSAMINE | CHEMBL335315 | N-(...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50240801(CHEMBL131967 | N-((2R,3R,4S,5S,6R)-3,4,5-trihydrox...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102884(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  1.05E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102884(8,9,10-Trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-...)
Affinity DataKi:  1.05E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50240801(CHEMBL131967 | N-((2R,3R,4S,5S,6R)-3,4,5-trihydrox...)
Affinity DataKi:  1.44E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102891(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-...)
Affinity DataKi:  3.70E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102890(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-...)
Affinity DataKi:  4.40E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102885(2,2,2-Trifluoro-N-(3,4,5-trihydroxy-6-hydroxymethy...)
Affinity DataKi:  7.10E+5nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102882(6-Hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol |...)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102888(2,3,4,5-Tetrahydroxy-6-hydroxymethyl-tetrahydro-py...)
Affinity DataKi:  3.10E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  7.40E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102892(8,9,10-Trihydroxy-2-thioxo-6-oxa-1,3-diaza-spiro[4...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102883(8,9,10-Trihydroxy-6-oxa-1,3-diaza-spiro[4.5]decane...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50102886(8,9,10-Trihydroxy-6-oxa-1,3-diaza-spiro[4.5]decane...)
Affinity DataKi:  1.15E+7nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed