Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50036960
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  7.14nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  204nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  281nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed