Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50011418
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  460nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  530nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50041119(2-(2-fluorophenyl)-6,7-methylenedioxyquinolin-4-on...)
Affinity DataIC50:  680nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106310(2,2-Dimethyl-propionic acid 6-(2-fluoro-phenyl)-8-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50012666(2-((E)-Styryl)-3H-quinazolin-4-one | 2-Styryl-3H-q...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM48563(2-phenyl-1H-quinolin-4-one | 2-phenyl-4-quinolone ...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106308(4-[6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106307(2-Phenyl-2,3-dihydro-1H-quinazolin-4-one | CHEMBL1...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106306(CHEMBL338626 | [6-(2-Fluoro-phenyl)-[1,3]dioxolo[4...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106311(6-(2-Fluoro-phenyl)-5H-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50041119(2-(2-fluorophenyl)-6,7-methylenedioxyquinolin-4-on...)
Affinity DataIC50:  3.90E+4nMAssay Description:Percent inhibition of colchicine binding(ICB) at 5 uM [3H]-colchicine concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106303(4-[6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106304(CHEMBL129338 | [6-(2-Fluoro-phenyl)-[1,3]dioxolo[4...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50044965(1-Methyl-2-phenyl-1H-quinolin-4-one | CHEMBL277048)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106305(2-Phenyl-3H-quinazolin-4-one | 2-phenyl-3,4-dihydr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerization.(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2'-fluorophenyl)-6-pyrolinyl-4-(1H)-quinolone |...)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of colchicine binding(ICB). Tubulin concentration was 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2'-fluorophenyl)-6-pyrolinyl-4-(1H)-quinolone |...)
Affinity DataIC50:  9.30E+4nMAssay Description:Inhibition of colchicine binding(ICB). [3H]-colchicine concentration was 5 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed