Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50011462
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106769(1-(2-{Bis-[3-(bis-{3-[bis-(3-amino-propyl)-amino]-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106770(2-(2-{Bis-[3-(bis-{3-[bis-(3-amino-propyl)-amino]-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106768(3-[[3-((3-{(2-Amino-ethyl)-[3-(bis-{3-[bis-(2-cyan...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106765(3-[[3-((3-{[2-(5-Amino-1,3-dioxo-1H,3H-benzo[de]is...)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106767(3-[[3-((3-{[3-(Bis-{3-[bis-(2-cyano-ethyl)-amino]-...)
Affinity DataIC50:  3.38E+4nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106764(3-[[3-((3-{[3-(Bis-{3-[bis-(2-cyano-ethyl)-amino]-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University San Pablo-Ceu

Curated by ChEMBL
LigandPNGBDBM50106766(3-[[3-((3-{[3-(Bis-{3-[bis-(2-cyano-ethyl)-amino]-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of lck catalytic domain expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed