Compile Data Set for Download or QSAR
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Found 21 Enz. Inhib. hit(s) with all data for entry = 5335
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85836([N-benzol]h alpha-CGRP8-37)
Affinity DataKi:  0.0720nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85837(h alpha-CGRP)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85837(h alpha-CGRP)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85836([N-benzol]h alpha-CGRP8-37)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85840([N-acetyl]h alpha-CGRP8-37)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85840([N-acetyl]h alpha-CGRP8-37)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85834([Pro14]h alpha-CGRP)
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50000743(CHEMBL525571 | [Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Se...)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50000743(CHEMBL525571 | [Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Se...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85834([Pro14]h alpha-CGRP)
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85843([D-Pen2,7]h alpha-CGRP)
Affinity DataKi:  15.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85841(Adrenomedullin)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85843([D-Pen2,7]h alpha-CGRP)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85835([Cys(ACM)2,7]h alpha-CGRP)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85838([Cha37]h alpha-CGRP8-37)
Affinity DataKi:  32.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85838([Cha37]h alpha-CGRP8-37)
Affinity DataKi:  37.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85835([Cys(ACM)2,7]h alpha-CGRP)
Affinity DataKi:  38.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85839([Pro34,Phe35]h alpha-CGRP27-37)
Affinity DataKi:  50.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85839([Pro34,Phe35]h alpha-CGRP27-37)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCalcitonin gene-related peptide type 1 receptor(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85842([Ala37]h alpha-CGRP8-37)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor activity-modifying protein 1(PIG)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM85842([Ala37]h alpha-CGRP8-37)
Affinity DataKi:  1.02E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed