Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50011524
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  800nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107543(4-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  2.20E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107542(3-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  1.30E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107543(4-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  3.00E+3nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50: >7.80E+4nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107541(2-Ethoxy-3-[4-methoxy-3-(4-trifluoromethyl-benzylc...)
Affinity DataEC50:  1.60E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107544(3-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  2.90E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107546(2-(3-((4-(trifluoromethyl)benzyl)carbamoyl)-4-meth...)
Affinity DataEC50:  40nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107545(3-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  240nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107548(2-Ethyl-2-[4-methoxy-3-(4-trifluoromethyl-benzylca...)
Affinity DataEC50:  2.80E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50: >1.37E+5nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  1.00E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107547(2-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  290nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107546(2-(3-((4-(trifluoromethyl)benzyl)carbamoyl)-4-meth...)
Affinity DataEC50:  400nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107551(2-Methoxy-3-[4-methoxy-3-(4-trifluoromethyl-benzyl...)
Affinity DataEC50:  230nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107550(2-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  360nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107549(2-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  2.50E+3nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107549(2-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)...)
Affinity DataEC50:  1.00E+3nMAssay Description:Transactivation of human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50107541(2-Ethoxy-3-[4-methoxy-3-(4-trifluoromethyl-benzylc...)
Affinity DataEC50:  2.80E+3nMAssay Description:Concentration of compound that affords half-maximum transactivation of human Peroxisome proliferator activated receptor gamma in CHO-K1 cells was det...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed