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Found 18 Enz. Inhib. hit(s) with all data for entry = 50011664
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50010960((E)-7-Phenyl-7-pyridin-3-yl-hept-6-enoic acid | 7-...)
Affinity DataIC50:  0.890nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109140(5-[1-Phenyl-1-pyridin-3-yl-meth-(Z)-ylideneaminoox...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109134(5-[1-Pyridin-3-yl-1-{3-[(3-pyridin-3-yl-1H-pyrrolo...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109124(5-[1-(3-{[4-(2-Methyl-imidazo[4,5-c]pyridin-1-ylme...)
Affinity DataIC50:  1.80nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109128(5-[1-Pyridin-3-yl-1-{4-[(3-pyridin-3-yl-1H-pyrrolo...)
Affinity DataIC50:  3.60nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109132(5-[1-(3-{[4-(2-Methyl-imidazo[4,5-c]pyridin-1-ylme...)
Affinity DataIC50:  4.70nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50404012(CHEMBL2111765)
Affinity DataIC50:  5.80nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109137(5-[1-Pyridin-3-yl-1-{3-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109126(5-[1-Pyridin-3-yl-1-{4-[(2-pyridin-3-yl-thiazolidi...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109131(5-[1-Pyridin-3-yl-1-{3-[(2-pyridin-3-yl-thiazolidi...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109135(5-[1-Pyridin-3-yl-1-{4-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109130(5-[1-Pyridin-3-yl-1-{3-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50:  52nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109127(5-[(3-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  65nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109129(5-[(4-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109136(5-[1-Pyridin-3-yl-1-{4-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109125(5-[1-Pyridin-3-yl-1-{3-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50:  88nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109133(5-[1-Pyridin-3-yl-1-{2-[4-(2-pyridin-3-yl-thiazoli...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed