Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 50035274
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110382(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  0.540nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110393(5-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  0.600nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110394(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  0.950nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110387(4-{2-[(S)-5-((S)-2,3-Dihydro-benzofuran-5-sulfonyl...)
Affinity DataKi:  2.5nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110389(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  3.20nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110393(5-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  5.90nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110389(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  6.20nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110374(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  7.60nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110391(4-[3-((S)-3-Benzenesulfonylamino-2-oxo-azepan-1-yl...)
Affinity DataKi:  8.30nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110386(4-{3-[(S)-3-(2,5-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  9nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110387(4-{2-[(S)-5-((S)-2,3-Dihydro-benzofuran-5-sulfonyl...)
Affinity DataKi:  11nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110392(4-{3-[(S)-3-(3,4-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  12nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110375(4-{3-[(S)-3-(Naphthalene-2-sulfonylamino)-2-oxo-az...)
Affinity DataKi:  12nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110392(4-{3-[(S)-3-(3,4-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  13nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110379(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  14nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110394(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  16nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110382(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  18nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110385(4-[2-Oxo-3-((S)-2-oxo-3-phenylmethanesulfonylamino...)
Affinity DataKi:  19nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110391(4-[3-((S)-3-Benzenesulfonylamino-2-oxo-azepan-1-yl...)
Affinity DataKi:  19nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110379(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  20nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110397(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  24nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110374(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  30nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110386(4-{3-[(S)-3-(2,5-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  35nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110382(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  40nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110381(2,3-Dihydro-benzofuran-5-sulfonic acid {(S)-1-[3-(...)
Affinity DataKi:  40nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110387(4-{2-[(S)-5-((S)-2,3-Dihydro-benzofuran-5-sulfonyl...)
Affinity DataKi:  49nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110393(5-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110377(2,3-Dihydro-benzofuran-5-sulfonic acid {(S)-1-[3-(...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110396(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  61nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110388(4-[3-((S)-3-Benzenesulfonylamino-2-oxo-azepan-1-yl...)
Affinity DataKi:  71nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110373(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  81nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110385(4-[2-Oxo-3-((S)-2-oxo-3-phenylmethanesulfonylamino...)
Affinity DataKi:  85nMAssay Description:Inhibitory constant against trypsin determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110384(4-{3-[(S)-3-(3,4-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  86nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110394(P1 argininal derivative | [amino({[(4S)-4-carboxy-...)
Affinity DataKi:  93nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110378(CHEMBL350262 | N-{(S)-1-[3-(6-Amino-2-methyl-pyrid...)
Affinity DataKi:  93nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110375(4-{3-[(S)-3-(Naphthalene-2-sulfonylamino)-2-oxo-az...)
Affinity DataKi:  164nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110376(4-{3-[(S)-3-(2,5-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi:  167nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110390(CHEMBL350117 | N-{(S)-1-[3-(4-Amino-cyclohexyl)-2-...)
Affinity DataKi:  195nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110373(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi:  240nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110395(2,3-Dihydro-benzofuran-5-sulfonic acid {(S)-1-[3-(...)
Affinity DataKi:  283nMAssay Description:Inhibitory constant against human thrombin (FIIa) determined in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110385(4-[2-Oxo-3-((S)-2-oxo-3-phenylmethanesulfonylamino...)
Affinity DataKi:  315nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110392(4-{3-[(S)-3-(3,4-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110391(4-[3-((S)-3-Benzenesulfonylamino-2-oxo-azepan-1-yl...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110381(2,3-Dihydro-benzofuran-5-sulfonic acid {(S)-1-[3-(...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110388(4-[3-((S)-3-Benzenesulfonylamino-2-oxo-azepan-1-yl...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110374(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110375(4-{3-[(S)-3-(Naphthalene-2-sulfonylamino)-2-oxo-az...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110384(4-{3-[(S)-3-(3,4-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110386(4-{3-[(S)-3-(2,5-Dimethoxy-benzenesulfonylamino)-2...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50110379(4-{3-[(S)-3-(2,3-Dihydro-benzofuran-5-sulfonylamin...)
Affinity DataKi: >338nMAssay Description:Inhibitory constant against human Coagulation factor Xa determined in VitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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