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Found 24 Enz. Inhib. hit(s) with all data for entry = 50012125
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  8nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50403914(CHEMBL2113711)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114973(CHEMBL51542 | N-(4-{[(Naphthalen-2-ylmethyl)-amino...)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114977(CHEMBL51884 | Naphthalene-1-sulfonic acid (4-{[(1,...)
Affinity DataKi:  11nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114979(CHEMBL415926 | Naphthalene-2-sulfonic acid (4-{[(1...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114976(2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114978(CHEMBL299295 | Naphthalene-1-sulfonic acid (4-{[2-...)
Affinity DataKi:  17nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  18nMAssay Description:Functional response of NPY to inhibit forskolin-stimulated cAMP in cells stably transfected with rat Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114981(CHEMBL51874 | N-(4-{[(Naphthalen-1-ylmethyl)-amino...)
Affinity DataKi:  26nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114980(2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl...)
Affinity DataKi:  28nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  63nMAssay Description:Binding affinity of the compound against cloned human Dopamine receptor D2 was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  100nMAssay Description:Bnding affinity of the compound against cloned human Alpha-2C adrenergic receptor was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114975(CHEMBL48777 | Naphthalene-2-sulfonic acid {6-[(nap...)
Affinity DataKi:  123nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114978(CHEMBL299295 | Naphthalene-1-sulfonic acid (4-{[2-...)
Affinity DataKi:  3.24E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114977(CHEMBL51884 | Naphthalene-1-sulfonic acid (4-{[(1,...)
Affinity DataKi:  3.55E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114979(CHEMBL415926 | Naphthalene-2-sulfonic acid (4-{[(1...)
Affinity DataKi:  5.55E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114975(CHEMBL48777 | Naphthalene-2-sulfonic acid {6-[(nap...)
Affinity DataKi:  7.30E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114973(CHEMBL51542 | N-(4-{[(Naphthalen-2-ylmethyl)-amino...)
Affinity DataKi:  1.30E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114981(CHEMBL51874 | N-(4-{[(Naphthalen-1-ylmethyl)-amino...)
Affinity DataKi:  1.45E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  1.60E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50403914(CHEMBL2113711)
Affinity DataKi:  1.72E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataKi:  2.20E+4nMAssay Description:Functional response of NPY to inhibit forskolin-stimulated cAMP in cells stably transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114976(2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl...)
Affinity DataKi:  2.37E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114980(2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl...)
Affinity DataKi:  4.87E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed