Compile Data Set for Download or QSAR
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Found 34 Enz. Inhib. hit(s) with all data for entry = 50035235
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114997(4-(4-Chloro-3-methyl-phenyl)-3-(4-chloro-phenyl)-3...)
Affinity DataKi:  24nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114997(4-(4-Chloro-3-methyl-phenyl)-3-(4-chloro-phenyl)-3...)
Affinity DataKi:  24nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115000(4-(4-Chloro-phenyl)-3-(3-trifluoromethyl-phenyl)-3...)
Affinity DataKi:  26nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115005(4-(4-Chloro-phenyl)-3-(2-fluoro-phenyl)-3H-thiazol...)
Affinity DataKi:  36nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114996(3-(4-Chloro-3-methyl-phenyl)-4-(2,6-difluoro-pheny...)
Affinity DataKi:  48nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114996(3-(4-Chloro-3-methyl-phenyl)-4-(2,6-difluoro-pheny...)
Affinity DataKi:  48nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115001(4-(4-Bromo-phenyl)-3-(3-trifluoromethyl-phenyl)-3H...)
Affinity DataKi:  67nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115001(4-(4-Bromo-phenyl)-3-(3-trifluoromethyl-phenyl)-3H...)
Affinity DataKi:  71nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114996(3-(4-Chloro-3-methyl-phenyl)-4-(2,6-difluoro-pheny...)
Affinity DataKi:  86nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115000(4-(4-Chloro-phenyl)-3-(3-trifluoromethyl-phenyl)-3...)
Affinity DataKi:  86nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114997(4-(4-Chloro-3-methyl-phenyl)-3-(4-chloro-phenyl)-3...)
Affinity DataKi:  99nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  108nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114999(3-(4-Chloro-phenyl)-4-p-tolyl-3H-thiazol-(2E)-ylid...)
Affinity DataKi:  124nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114999(3-(4-Chloro-phenyl)-4-p-tolyl-3H-thiazol-(2E)-ylid...)
Affinity DataKi:  124nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115001(4-(4-Bromo-phenyl)-3-(3-trifluoromethyl-phenyl)-3H...)
Affinity DataKi:  140nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115003(4-(4-Chloro-phenyl)-3-(2,4-dichloro-phenyl)-3H-thi...)
Affinity DataKi:  141nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  155nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115005(4-(4-Chloro-phenyl)-3-(2-fluoro-phenyl)-3H-thiazol...)
Affinity DataKi:  189nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114997(4-(4-Chloro-3-methyl-phenyl)-3-(4-chloro-phenyl)-3...)
Affinity DataKi:  225nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  274nMAssay Description:Compound was tested for the inhibition of [3H]DA reuptake into rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115000(4-(4-Chloro-phenyl)-3-(3-trifluoromethyl-phenyl)-3...)
Affinity DataKi:  398nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114998(4-(4-Chloro-phenyl)-3-(2-morpholin-4-yl-phenyl)-3H...)
Affinity DataKi:  424nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114996(3-(4-Chloro-3-methyl-phenyl)-4-(2,6-difluoro-pheny...)
Affinity DataKi:  433nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115003(4-(4-Chloro-phenyl)-3-(2,4-dichloro-phenyl)-3H-thi...)
Affinity DataKi:  533nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114999(3-(4-Chloro-phenyl)-4-p-tolyl-3H-thiazol-(2E)-ylid...)
Affinity DataKi:  801nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115003(4-(4-Chloro-phenyl)-3-(2,4-dichloro-phenyl)-3H-thi...)
Affinity DataKi:  843nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115007(2,3-Diphenyl-pyrazine | CHEMBL48222)
Affinity DataKi: >1.00E+3nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115004(3-Methyl-4,5-diphenyl-3H-pyridin-2-one | CHEMBL499...)
Affinity DataKi: >1.00E+3nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115005(4-(4-Chloro-phenyl)-3-(2-fluoro-phenyl)-3H-thiazol...)
Affinity DataKi:  1.41E+3nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115002(2-Methyl-4,5-diphenyl-4,5-dihydro-thiazole | CHEMB...)
Affinity DataKi:  2.28E+3nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114999(3-(4-Chloro-phenyl)-4-p-tolyl-3H-thiazol-(2E)-ylid...)
Affinity DataKi:  2.62E+3nMAssay Description:Compound was tested for the inhibition of serotonin [3H]SER reuptake into rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50115006(3-(4-Chloro-phenyl)-4-phenyl-4H-[1,2,4]oxadiazol-5...)
Affinity DataKi:  9.18E+3nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114998(4-(4-Chloro-phenyl)-3-(2-morpholin-4-yl-phenyl)-3H...)
Affinity DataKi:  2.21E+4nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50114998(4-(4-Chloro-phenyl)-3-(2-morpholin-4-yl-phenyl)-3H...)
Affinity DataKi:  4.20E+4nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed