Compile Data Set for Download or QSAR
maximum 50k data
Found 162 Enz. Inhib. hit(s) with all data for entry = 50041046
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220468(CHEMBL61120)
Affinity DataKi:  0.501nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220419(CHEMBL63125)
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139308((R)-2-Amino-1-{4-[3-(4-cyclopropanecarbonyl-phenox...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220473(CHEMBL305144)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220430(CHEMBL302829)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220467(CHEMBL62421)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220430(CHEMBL302829)
Affinity DataKi:  1.95nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220417(CHEMBL64406)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220422(CHEMBL60401)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220449(CHEMBL60837)
Affinity DataKi:  2.40nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220428(CHEMBL418666)
Affinity DataKi:  2.5nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220434(CHEMBL291821)
Affinity DataKi:  4nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220457(CHEMBL60143)
Affinity DataKi:  4nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220459(CHEMBL62596)
Affinity DataKi:  4.40nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220439(CHEMBL64059)
Affinity DataKi:  4.60nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220437(CHEMBL61792)
Affinity DataKi:  4.60nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220433(CHEMBL60435)
Affinity DataKi:  4.70nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220461(CHEMBL59733)
Affinity DataKi:  5.80nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220427(CHEMBL64608)
Affinity DataKi:  6.5nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220471(CHEMBL62660)
Affinity DataKi:  7.10nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220470(CHEMBL293033)
Affinity DataKi:  8.5nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220460(CHEMBL304888)
Affinity DataKi:  8.70nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220426(CHEMBL61288)
Affinity DataKi:  8.90nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220472(CHEMBL64321)
Affinity DataKi:  9.10nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220464(CHEMBL62808)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220438(CHEMBL59931)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220436(CHEMBL64896)
Affinity DataKi:  13nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220418(CHEMBL59870)
Affinity DataKi:  14nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220440(CHEMBL60598)
Affinity DataKi:  15nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220462(CHEMBL303369)
Affinity DataKi:  17nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220431(CHEMBL62804)
Affinity DataKi:  20nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220450(CHEMBL62903)
Affinity DataKi:  23nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220452(CHEMBL60559)
Affinity DataKi:  23nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220455(CHEMBL434785)
Affinity DataKi:  26nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220425(CHEMBL302468)
Affinity DataKi:  28nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220454(CHEMBL64124)
Affinity DataKi:  29nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220429(CHEMBL305371)
Affinity DataKi:  30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220442(CHEMBL64461)
Affinity DataKi:  30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220456(CHEMBL417215)
Affinity DataKi:  30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220423(CHEMBL423666)
Affinity DataKi:  43nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220421(CHEMBL62050)
Affinity DataKi:  44nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220469(CHEMBL62716)
Affinity DataKi:  52nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220432(CHEMBL62266)
Affinity DataKi:  54nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220435(CHEMBL62741)
Affinity DataKi:  62nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220441(CHEMBL294087)
Affinity DataKi:  76nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220465(CHEMBL62592)
Affinity DataKi:  79nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220453(CHEMBL312958)
Affinity DataKi:  98nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220420(CHEMBL63112)
Affinity DataKi:  112nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220451(CHEMBL64120)
Affinity DataKi:  120nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220424(CHEMBL60189)
Affinity DataKi:  132nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 162 total ) | Next | Last >>
Jump to: