Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50012375
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118202(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118204(6-(4-benzoylphenylcarbonyloxy)-8-(tert-butyl)-12,1...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118194(8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-t...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118201(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-12,17-dihydr...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118203(8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-6-[4-(...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118195(3'-(tert-butyl)-4,9',14'-trihydroxy-2-methoxy-10'-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118196(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-9,12,17-trih...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118200(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118205(3'-(tert-butyl)-4,9'-dihydroxy-2-methoxy-10'-methy...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118193(3'-(tert-butyl)-4,4',9'-trihydroxy-2-methoxy-10'-m...)
Affinity DataKi:  9.90E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118197(3'-(tert-butyl)-4,4',9',14'-tetrahydroxy-2-methoxy...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118198(3'-(tert-butyl)-4,4',14'-trihydroxy-2-methoxy-10'-...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118199(9-tert-Butyl-8,9-dihydroxy-dihydro-furo[2,3-b]furo...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed