Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50012409
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118655(CHEMBL432649 | Ca-pYEEIE)
Affinity DataIC50:  42nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118655(CHEMBL432649 | Ca-pYEEIE)
Affinity DataIC50:  64nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118660(CHEMBL90976 | Cm-pYEEIE)
Affinity DataIC50:  81nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118655(CHEMBL432649 | Ca-pYEEIE)
Affinity DataIC50:  84nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118660(CHEMBL90976 | Cm-pYEEIE)
Affinity DataIC50:  90nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118660(CHEMBL90976 | Cm-pYEEIE)
Affinity DataIC50:  100nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  1.10E+3nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  1.30E+3nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  2.00E+3nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118658(Ac-YAEIE | CHEMBL90294)
Affinity DataIC50:  3.80E+3nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118658(Ac-YAEIE | CHEMBL90294)
Affinity DataIC50:  7.00E+3nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118658(Ac-YAEIE | CHEMBL90294)
Affinity DataIC50:  1.10E+4nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118654(CHEMBL328034 | Ca-DOPA-EEIE)
Affinity DataIC50:  1.80E+4nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118659(CHEMBL327820 | Ca-YEEIE)
Affinity DataIC50:  2.70E+4nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118654(CHEMBL328034 | Ca-DOPA-EEIE)
Affinity DataIC50:  3.30E+4nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118659(CHEMBL327820 | Ca-YEEIE)
Affinity DataIC50:  4.50E+4nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118659(CHEMBL327820 | Ca-YEEIE)
Affinity DataIC50:  5.40E+4nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118654(CHEMBL328034 | Ca-DOPA-EEIE)
Affinity DataIC50:  5.50E+4nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118656(CHEMBL430902 | CM-DOPA-EEIE)
Affinity DataIC50:  5.80E+4nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118656(CHEMBL430902 | CM-DOPA-EEIE)
Affinity DataIC50:  6.50E+4nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118656(CHEMBL430902 | CM-DOPA-EEIE)
Affinity DataIC50:  7.70E+4nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118661(AC-DOPA-EEE | CHEMBL2370170)
Affinity DataIC50:  1.20E+5nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118661(AC-DOPA-EEE | CHEMBL2370170)
Affinity DataIC50:  1.20E+5nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118653(Ac-YEEIE | CHEMBL329886)
Affinity DataIC50: >2.00E+5nMAssay Description:Affinity for GST- Src-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118661(AC-DOPA-EEE | CHEMBL2370170)
Affinity DataIC50: >2.00E+5nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118653(Ac-YEEIE | CHEMBL329886)
Affinity DataIC50: >2.00E+5nMAssay Description:Affinity for GST-Lck-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Mogam Biotechnology Research Institute

Curated by ChEMBL
LigandPNGBDBM50118653(Ac-YEEIE | CHEMBL329886)
Affinity DataIC50: >2.00E+5nMAssay Description:Affinity for GST-Fyn-SH2 domain in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed