Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50012411
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50403954(CHEMBL2112366)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118664(5-{3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl...)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118666(3-[2-Methoxy-5-(5-trifluoromethyl-tetrazol-1-yl)-p...)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118667(7-(1H-Imidazol-4-ylmethyl)-3-[2-methoxy-5-(5-trifl...)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50403953(CHEMBL2112368)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118671(3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-1...)
Affinity DataIC50:  0.350nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118670(3-(2-Methoxy-5-trifluoromethoxy-phenyl)-6-phenyl-7...)
Affinity DataIC50:  0.890nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118662(3-(2-Methoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4....)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118663(3-(2-Methoxy-phenyl)-6-phenyl-1-oxa-7-aza-spiro[4....)
Affinity DataIC50:  49nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50403952(CHEMBL2112367)
Affinity DataIC50:  133nMAssay Description:Displacement of [125I]-labeled substance P from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed