Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 50035257
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataKi:  2nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataKi:  125nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM11464((2S,3S)-2-amino-3-methyl-1-(1,3-thiazolidin-3-yl)p...)
Affinity DataKi:  126nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118940((S)-1-((S)-2-Amino-propionyl)-pyrrolidine-2-carbon...)
Affinity DataKi:  200nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118943((2S,3S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)pentan...)
Affinity DataKi:  218nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118934((S)-2-Amino-1-thiazolidin-3-yl-propane-1-thione | ...)
Affinity DataKi:  277nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118946((S)-2-Amino-1-pyrrolidin-1-yl-propane-1-thione | C...)
Affinity DataKi:  1.43E+3nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118934((S)-2-Amino-1-thiazolidin-3-yl-propane-1-thione | ...)
Affinity DataKi:  7.88E+3nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM11464((2S,3S)-2-amino-3-methyl-1-(1,3-thiazolidin-3-yl)p...)
Affinity DataKi:  8.17E+3nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118943((2S,3S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)pentan...)
Affinity DataKi:  2.47E+4nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118946((S)-2-Amino-1-pyrrolidin-1-yl-propane-1-thione | C...)
Affinity DataKi:  4.76E+4nMAssay Description:Inhibition of Dipeptidyl Peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118950((3S)-4-oxo-4-piperidin-1-ylbutane-1,3-diamine | (S...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118935(2-Amino-3-(1H-imidazol-4-yl)-1-piperidin-1-yl-prop...)
Affinity DataIC50:  328nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118945(2,5-Diamino-1-piperidin-1-yl-pentan-1-one | CHEMBL...)
Affinity DataIC50:  450nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118942(2-Amino-3-(1H-imidazol-4-yl)-1-pyrrolidin-1-yl-pro...)
Affinity DataIC50:  1.16E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118953(2,6-Diamino-1-piperidin-1-yl-hexan-1-one | CHEMBL9...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118933((S)-2,3-Diamino-1-piperidin-1-yl-propan-1-one | CH...)
Affinity DataIC50:  1.84E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118941(CHEMBL94955 | [5-Amino-1-(piperidine-1-carbonyl)-p...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50178428((S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)butan-1-on...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118943((2S,3S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)pentan...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118938(2-Cyclohexylamino-1-piperidin-1-yl-propan-1-one | ...)
Affinity DataIC50:  9.90E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118947(2,6-Diamino-1-pyrrolidin-1-yl-hexan-1-one | CHEMBL...)
Affinity DataIC50:  9.90E+3nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118937(2-Amino-3-(4-hydroxy-phenyl)-1-pyrrolidin-1-yl-pro...)
Affinity DataIC50:  1.40E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50228295((S)-pyrrolidin-1-yl(pyrrolidin-2-yl)methanone | CH...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118932((S)-2-Amino-3-cyclohexyl-1-pyrrolidin-1-yl-propan-...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118939(2-Amino-3-phenyl-1-pyrrolidin-1-yl-propan-1-one | ...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118942(2-Amino-3-(1H-imidazol-4-yl)-1-pyrrolidin-1-yl-pro...)
Affinity DataIC50:  2.32E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118947(2,6-Diamino-1-pyrrolidin-1-yl-hexan-1-one | CHEMBL...)
Affinity DataIC50:  3.90E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50243406((S)-2-amino-1-(pyrrolidin-1-yl)propan-1-one | CHEM...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Dipeptidyl Peptidase II (Quiescent cell proline peptidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118932((S)-2-Amino-3-cyclohexyl-1-pyrrolidin-1-yl-propan-...)
Affinity DataIC50:  4.20E+4nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118936(2-Amino-3-methyl-1-piperidin-1-yl-pentan-1-one | 3...)
Affinity DataIC50:  6.20E+4nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118949(2-Amino-3-hydroxy-1-pyrrolidin-1-yl-propan-1-one |...)
Affinity DataIC50:  6.50E+4nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118936(2-Amino-3-methyl-1-piperidin-1-yl-pentan-1-one | 3...)
Affinity DataIC50:  6.70E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118939(2-Amino-3-phenyl-1-pyrrolidin-1-yl-propan-1-one | ...)
Affinity DataIC50:  7.90E+4nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118940((S)-1-((S)-2-Amino-propionyl)-pyrrolidine-2-carbon...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibitory activity against Dipeptidyl Peptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118943((2S,3S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)pentan...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50243412((S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanoic acid...)
Affinity DataIC50:  1.22E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118941(CHEMBL94955 | [5-Amino-1-(piperidine-1-carbonyl)-p...)
Affinity DataIC50:  1.35E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118937(2-Amino-3-(4-hydroxy-phenyl)-1-pyrrolidin-1-yl-pro...)
Affinity DataIC50:  1.50E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118948(3-Amino-4-oxo-4-pyrrolidin-1-yl-butyramide | CHEMB...)
Affinity DataIC50:  1.52E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50243406((S)-2-amino-1-(pyrrolidin-1-yl)propan-1-one | CHEM...)
Affinity DataIC50:  1.79E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118948(3-Amino-4-oxo-4-pyrrolidin-1-yl-butyramide | CHEMB...)
Affinity DataIC50:  1.88E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118949(2-Amino-3-hydroxy-1-pyrrolidin-1-yl-propan-1-one |...)
Affinity DataIC50:  1.90E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118935(2-Amino-3-(1H-imidazol-4-yl)-1-piperidin-1-yl-prop...)
Affinity DataIC50:  2.13E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118938(2-Cyclohexylamino-1-piperidin-1-yl-propan-1-one | ...)
Affinity DataIC50:  2.17E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50178428((S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)butan-1-on...)
Affinity DataIC50:  2.23E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118953(2,6-Diamino-1-piperidin-1-yl-hexan-1-one | CHEMBL9...)
Affinity DataIC50:  2.47E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50228295((S)-pyrrolidin-1-yl(pyrrolidin-2-yl)methanone | CH...)
Affinity DataIC50: >5.00E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50243412((S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanoic acid...)
Affinity DataIC50: >5.00E+5nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase II.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118945(2,5-Diamino-1-piperidin-1-yl-pentan-1-one | CHEMBL...)
Affinity DataIC50: >5.00E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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