TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 6.70E+4nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair