Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50012778
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataKi:  2.90nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122722(9-Butyl-5-(piperidin-4-ylmethoxy)-1,2,3,4-tetrahyd...)
Affinity DataKi:  10nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122721(6-(1-Ethyl-piperidin-4-ylmethoxy)-8,9,10,11-tetrah...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122719(9-Pentyl-5-(piperidin-4-ylmethoxy)-1,2,3,4-tetrahy...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122718(6-(1-Propyl-piperidin-4-ylmethoxy)-8,9,10,11-tetra...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122723(9-Ethyl-5-(piperidin-4-ylmethoxy)-1,2,3,4-tetrahyd...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122720(6-(1-Butyl-piperidin-4-ylmethoxy)-8,9,10,11-tetrah...)
Affinity DataKi:  16nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université

Curated by ChEMBL
LigandPNGBDBM50122717(9-Methyl-5-(piperidin-4-ylmethoxy)-1,2,3,4-tetrahy...)
Affinity DataKi:  80nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  0.560nMAssay Description:Ability to displace [3H]GR-113808 from mouse 5-hydroxytryptamine 4 receptor in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  200nMAssay Description:Ability to displace [3H]5-HT from 5-hydroxytryptamine 2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  3.20E+3nMAssay Description:Ability to displace [3H]AVP from vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  3.40E+3nMAssay Description:Ability to displace [3H]mesulergine from 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  3.40E+3nMAssay Description:Ability to displace [3H]YM-0915 from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  5.00E+3nMAssay Description:Ability to displace [3H]-ketanserin from 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  9.10E+3nMAssay Description:Ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Sus scrofa)
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  1.10E+4nMAssay Description:Ability to displace [3H]AVP from Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Mus musculus (Mouse))
Université

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to displace [3H]SCH-23390 from Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed