Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50012818
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50097626(1-(3-Carbamimidoyl-phenyl)-1H-tetrazole-5-carboxyl...)
Affinity DataKi:  0.0370nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123033(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123037(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  0.390nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123038(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123035(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123039(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123043(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  3nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123041(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123036(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50097626(1-(3-Carbamimidoyl-phenyl)-1H-tetrazole-5-carboxyl...)
Affinity DataKi:  6.40nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123040(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  8nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123034(1-(4-Methoxy-phenyl)-1H-tetrazole-5-carboxylic aci...)
Affinity DataKi:  8nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123042(1-(3-Aminomethyl-phenyl)-1H-tetrazole-5-carboxylic...)
Affinity DataKi:  13nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123031(1-(3-Amino-4-methoxy-phenyl)-1H-tetrazole-5-carbox...)
Affinity DataKi:  19nMAssay Description:Inhibition of human purified factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123042(1-(3-Aminomethyl-phenyl)-1H-tetrazole-5-carboxylic...)
Affinity DataKi:  69nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50097626(1-(3-Carbamimidoyl-phenyl)-1H-tetrazole-5-carboxyl...)
Affinity DataKi:  300nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123037(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  400nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123033(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  600nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123043(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123038(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123034(1-(4-Methoxy-phenyl)-1H-tetrazole-5-carboxylic aci...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123031(1-(3-Amino-4-methoxy-phenyl)-1H-tetrazole-5-carbox...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123038(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123037(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123041(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123039(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123036(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123040(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123043(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123036(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi: >1.60E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123041(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123031(1-(3-Amino-4-methoxy-phenyl)-1H-tetrazole-5-carbox...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123033(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi: >5.20E+3nMAssay Description:Inhibitory constant against trypsin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123040(1-(3-Amino-4-chloro-phenyl)-1H-tetrazole-5-carboxy...)
Affinity DataKi:  7.90E+3nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123034(1-(4-Methoxy-phenyl)-1H-tetrazole-5-carboxylic aci...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123039(1-(3-Amino-benzo[d]isoxazol-5-yl)-1H-tetrazole-5-c...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50123042(1-(3-Aminomethyl-phenyl)-1H-tetrazole-5-carboxylic...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibitory constant against thrombin using human purified enzymesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed