Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50012892
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123937(4-[8-Benzyl-17-{1-[1-(carbamoylmethyl-carbamoyl)-2...)
Affinity DataIC50:  440nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123939(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataIC50:  455nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123940(CHEMBL414177 | c[Gly-Pro-D-Nal(2')-Arg-Trp-Glu]-Va...)
Affinity DataIC50:  637nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(CHEMBL413177 | c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Va...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123946(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataIC50:  8.20E+3nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123936(19-Benzyl-16-(3-guanidino-propyl)-13-(1H-indol-3-y...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(CHEMBL413177 | c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Va...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123936(19-Benzyl-16-(3-guanidino-propyl)-13-(1H-indol-3-y...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123945(CHEMBL430267 | c[6-Ahx-His-D-phe-Arg-Trp-Glu]-Val-...)
Affinity DataEC50:  23nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123948(CHEMBL265804 | c[beta-Ala-His-D-phe-Arg-Trp-Glu]-V...)
Affinity DataEC50:  31nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123947(CHEMBL404931 | c[6-Ahx-His-phe-Arg-Trp-Glu]-Val-Va...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123946(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123949(CHEMBL406614 | c[gamma-Abu-His-D-Nal(2')-Arg-Trp-G...)
Affinity DataEC50:  23nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123940(CHEMBL414177 | c[Gly-Pro-D-Nal(2')-Arg-Trp-Glu]-Va...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123951(9-Benzyl-6-(3-guanidino-propyl)-12-(3H-imidazol-4-...)
Affinity DataEC50:  313nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123950(CHEMBL267755 | c[His-D-Nal(2')-Arg-Trp-Glu]-Val-Va...)
Affinity DataEC50:  60nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123942(CHEMBL269338 | c[beta-Ala-His-D-Nal(2')-Arg-Trp-Gl...)
Affinity DataEC50:  2nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123941(8-Benzyl-11-(3-guanidino-propyl)-5-(3H-imidazol-4-...)
Affinity DataEC50:  5.20E+3nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123939(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataEC50:  825nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123938(CHEMBL409760 | c[Gly-His-D-Nal(2')-Arg-Trp-Glu]-Va...)
Affinity DataEC50:  60nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123937(4-[8-Benzyl-17-{1-[1-(carbamoylmethyl-carbamoyl)-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123935(8-Benzyl-11-(3-guanidino-propyl)-5-(3H-imidazol-4-...)
Affinity DataEC50:  510nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50123944(9-Benzyl-6-(3-guanidino-propyl)-12-(3H-imidazol-4-...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed