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Found 35 Enz. Inhib. hit(s) with all data for entry = 50013037
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(CHEMBL13910 | N-[1-[2-(4-Butyryl-4-phenyl-piperidi...)
Affinity DataIC50:  3.10nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataIC50:  5.10nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(CHEMBL276012 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataIC50:  5.5nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(CHEMBL276301 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50:  32nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125751(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125745(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125745(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  510nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.5nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  28nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  2.20E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125746(1'-[3-(4-methoxyphenyl)-2-(1,2,3,4-tetrahydro-3-is...)
Affinity DataEC50:  40nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  4.40E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(CHEMBL276301 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  840nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  3.90E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(CHEMBL13910 | N-[1-[2-(4-Butyryl-4-phenyl-piperidi...)
Affinity DataEC50:  0.190nMAssay Description:In vitro inhibitory concentration against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  630nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.00E+4nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(CHEMBL276301 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  9.40E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  23nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(CHEMBL13910 | N-[1-[2-(4-Butyryl-4-phenyl-piperidi...)
Affinity DataEC50:  2.90nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  2.60E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(CHEMBL276012 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  2.70E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125746(1'-[3-(4-methoxyphenyl)-2-(1,2,3,4-tetrahydro-3-is...)
Affinity DataEC50:  220nMAssay Description:In vitro inhibitory concentration against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(CHEMBL276012 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  77nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(CHEMBL13910 | N-[1-[2-(4-Butyryl-4-phenyl-piperidi...)
Affinity DataEC50:  250nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125751(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  400nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(CHEMBL276012 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  3.90E+3nMAssay Description:In vitro effective concentration towards human Melanocortin-3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(CHEMBL276301 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  2.5nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.70E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(CHEMBL276012 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  3.80nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(CHEMBL13910 | N-[1-[2-(4-Butyryl-4-phenyl-piperidi...)
Affinity DataEC50:  2.10E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(CHEMBL276301 | N-[2-(4-Butyryl-4-phenyl-piperidin-...)
Affinity DataEC50:  7.00E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  0.350nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed