Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 50013042
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  31nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)
Affinity DataIC50:  430nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  600nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125833(3-(4-Fluoro-benzylidene)-1-hydroxy-5-isobutyl-3H-p...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409783(CHEMBL1626982 | CHEMBL2068710 | CHEMBL2068711 | CH...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409801(CHEMBL16525)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125793(4-(4-Cyclohexyl-phenyl)-2-hydroxy-4-oxo-but-2-enoi...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125822(1-Hydroxy-5-isobutyl-3-isobutylidene-3H-pyrazine-2...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Influenza B virus (B/Lee/40))
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409801(CHEMBL16525)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza B/Lee/40 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409805(CHEMBL278443)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409780(CHEMBL16239)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409787(CHEMBL16377)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409804(CHEMBL16453)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409802(CHEMBL277536)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409792(CHEMBL275631)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409789(CHEMBL16579)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409810(CHEMBL16887)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409785(CHEMBL280445)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409796(CHEMBL429766)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM33410(CHEMBL16755 | N-hydroxyisoquinolinedione, 2)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409793(CHEMBL280446)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409798(CHEMBL16233)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Influenza B virus (B/Lee/40))
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409787(CHEMBL16377)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza B/Lee/40 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409800(CHEMBL16336)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50115579((Z)-2-hydroxy-4-oxo-4-phenyl-but-2-enoic acid | 2-...)
Affinity DataIC50:  2.13E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409788(CHEMBL276316)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Influenza B virus (B/Lee/40))
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409802(CHEMBL277536)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza B/Lee/40 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Influenza B virus (B/Lee/40))
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409780(CHEMBL16239)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza B/Lee/40 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409779(CHEMBL16299)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50024265(CHEMBL2040641)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409803(CHEMBL1907704)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409782(CHEMBL279999)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409791(CHEMBL276589)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409797(CHEMBL275420)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409794(CHEMBL16313)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409784(CHEMBL16050)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409809(CHEMBL430143)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409781(CHEMBL16406)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409795(CHEMBL277284)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409807(CHEMBL16665)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza A/PR/8/34 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Influenza B virus (B/Lee/40))
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50409792(CHEMBL275631)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza B/Lee/40 RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125803(3-Hydroxy-1H-pteridine-2,4-dione | 3-hydroxypterid...)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM23987(2-hydroxy-1,2,3,4-tetrahydroisoquinolin-3-one | CH...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125805((3Z)-5-isobutyl-1-(methoxymethoxy)-3-(2-methylprop...)
Affinity DataIC50: >3.55E+5nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125809(3-(4-Fluoro-benzylidene)-5-isobutyl-3H-pyrazine-2,...)
Affinity DataIC50: >3.65E+5nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Roche Discovery Welwyn

Curated by ChEMBL
LigandPNGBDBM50125808(2-Hydroxy-isoindole-1,3-dione | 2-hydroxyisoindoli...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory concentration against cap-dependent endonuclease activity of influenza virus RNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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