Compile Data Set for Download or QSAR
maximum 50k data
Found 109 Enz. Inhib. hit(s) with all data for entry = 50041071
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  0.195nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50370569(A-349,821 | A-349821)
Affinity DataKi:  0.490nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222963(CHEMBL24863)
Affinity DataKi:  0.603nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222941(CHEMBL27501)
Affinity DataKi:  0.692nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223042(CHEMBL283313)
Affinity DataKi:  0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223041(CHEMBL280590)
Affinity DataKi:  0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223048(CHEMBL25519)
Affinity DataKi:  0.851nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222951(CHEMBL27933)
Affinity DataKi:  0.977nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223041(CHEMBL280590)
Affinity DataKi:  1nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222973(CHEMBL26880)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50370569(A-349,821 | A-349821)
Affinity DataKi:  1.70nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223042(CHEMBL283313)
Affinity DataKi:  2nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222950(CHEMBL279463)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222948(CHEMBL25342)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222964(CHEMBL27697)
Affinity DataKi:  2.40nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223048(CHEMBL25519)
Affinity DataKi:  2.80nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223038(CHEMBL433031)
Affinity DataKi:  2.80nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222957(CHEMBL2113223)
Affinity DataKi:  2.90nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222952(CHEMBL27665)
Affinity DataKi:  3nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222963(CHEMBL24863)
Affinity DataKi:  3nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222938(CHEMBL25685)
Affinity DataKi:  3.5nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222960(CHEMBL27444)
Affinity DataKi:  3.60nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223043(CHEMBL25205)
Affinity DataKi:  3.60nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223038(CHEMBL433031)
Affinity DataKi:  3.70nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222948(CHEMBL25342)
Affinity DataKi:  3.80nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222959(CHEMBL2113224)
Affinity DataKi:  3.90nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222951(CHEMBL27933)
Affinity DataKi:  4.20nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223044(CHEMBL436340)
Affinity DataKi:  4.40nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223043(CHEMBL25205)
Affinity DataKi:  4.70nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223040(CHEMBL281640)
Affinity DataKi:  4.80nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222969(CHEMBL282903)
Affinity DataKi:  5.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222941(CHEMBL27501)
Affinity DataKi:  5.10nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222965(CHEMBL2113222)
Affinity DataKi:  5.5nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222939(CHEMBL24468)
Affinity DataKi:  6.20nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222967(CHEMBL24198)
Affinity DataKi:  6.20nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222958(CHEMBL27339)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222961(CHEMBL27835)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222973(CHEMBL26880)
Affinity DataKi:  6.60nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222954(CHEMBL24865)
Affinity DataKi:  6.90nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222946(CHEMBL280895)
Affinity DataKi:  6.90nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222950(CHEMBL279463)
Affinity DataKi:  7.20nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217101(CHEMBL25688)
Affinity DataKi:  7.20nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223039(CHEMBL27209)
Affinity DataKi:  7.20nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222949(CHEMBL282062)
Affinity DataKi:  8.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222940(CHEMBL282685)
Affinity DataKi:  8.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223037(CHEMBL25501)
Affinity DataKi:  8.30nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222938(CHEMBL25685)
Affinity DataKi:  8.30nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50223039(CHEMBL27209)
Affinity DataKi:  8.70nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50222964(CHEMBL27697)
Affinity DataKi:  8.90nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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