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Found 18 Enz. Inhib. hit(s) with all data for entry = 50037242
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM20608(4-Hydroxytamoxifen | 4-Hydroxytamoxifen (9) | 4-[(...)
Affinity DataKi:  0.160nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM20608(4-Hydroxytamoxifen | 4-Hydroxytamoxifen (9) | 4-[(...)
Affinity DataKi:  0.25nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM20625(4-[(3E)-4-(4-hydroxyphenyl)hex-3-en-3-yl]phenol | ...)
Affinity DataKi:  0.490nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM20625(4-[(3E)-4-(4-hydroxyphenyl)hex-3-en-3-yl]phenol | ...)
Affinity DataKi:  0.630nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)
Affinity DataKi:  1.04nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)
Affinity DataKi:  1.39nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126767(7-Ethyl-4-methyl-9-[4-(2-piperidin-1-yl-ethoxy)-ph...)
Affinity DataKi:  8.69nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126766(7-(1-Hydroxy-ethyl)-4-methyl-9-[4-(2-piperidin-1-y...)
Affinity DataKi:  120nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126772(7-Isopropenyl-4-methyl-9-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi:  180nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126766(7-(1-Hydroxy-ethyl)-4-methyl-9-[4-(2-piperidin-1-y...)
Affinity DataKi:  190nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126767(7-Ethyl-4-methyl-9-[4-(2-piperidin-1-yl-ethoxy)-ph...)
Affinity DataKi:  190nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126770(7-(1,2-Dimethyl-propenyl)-4-methyl-9-[4-(2-piperid...)
Affinity DataKi:  200nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126770(7-(1,2-Dimethyl-propenyl)-4-methyl-9-[4-(2-piperid...)
Affinity DataKi:  210nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126772(7-Isopropenyl-4-methyl-9-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi:  290nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126768(1-{7-Hydroxy-5-methyl-10-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi:  490nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126771(1-{7-Hydroxy-5-methyl-10-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi:  630nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126768(1-{7-Hydroxy-5-methyl-10-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Signalgene

Curated by ChEMBL
LigandPNGBDBM50126771(1-{7-Hydroxy-5-methyl-10-[4-(2-piperidin-1-yl-etho...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro displacement of 0.5 nM [3H]17-beta-estradiol from human Estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed