Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50013162
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50075009(1-Ethyl-5-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  41nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127282(7-[(4-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  55nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127286(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  62nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127279(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50:  62nMAssay Description:In vitro inhibitiion of cytochrome P450 19A1 from human placental microsomes with 2.5 uM [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127285(5-Chloro-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-y...)
Affinity DataIC50:  63nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127281(7-[(4-Bromo-phenyl)-imidazol-1-yl-methyl]-1-ethyl-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127280(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  90nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127283(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  110nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127284(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50:  170nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127287(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127278(1-Ethyl-7-[(4-fluoro-phenyl)-[1,2,4]triazol-1-yl-m...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank