Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 50037139
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127626(5-(3',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  9.70nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127627(5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-...)
Affinity DataKi:  10.3nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  13.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127642(5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2....)
Affinity DataKi:  13.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  17.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  19.8nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127635(5-(4-Thiophen-3-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  20.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127624(5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-t...)
Affinity DataKi:  22.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127634(5-(4'-Methyl-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  22.7nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  32.4nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127638(5-(4'-Methoxy-biphenyl-4-ylmethylene)-3-aza-tricyc...)
Affinity DataKi:  39nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127628(5-(4-Pyrrol-1-yl-benzylidene)-3-aza-tricyclo[4.4.2...)
Affinity DataKi:  45.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  46nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  47nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  57nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127622(5-(4'-Methylamino-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  57.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127643(5-(3',5'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  61nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  71nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  73nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  89nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127642(5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2....)
Affinity DataKi:  98nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127643(5-(3',5'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  106nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  108nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127629(5-(4'-Iodo-biphenyl-4-ylmethylene)-3-aza-tricyclo[...)
Affinity DataKi:  114nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127635(5-(4-Thiophen-3-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  145nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127628(5-(4-Pyrrol-1-yl-benzylidene)-3-aza-tricyclo[4.4.2...)
Affinity DataKi:  149nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  155nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  155nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  165nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  179nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127624(5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-t...)
Affinity DataKi:  200nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  213nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127634(5-(4'-Methyl-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  214nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127626(5-(3',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  236nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127626(5-(3',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  239nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127642(5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2....)
Affinity DataKi:  248nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127635(5-(4-Thiophen-3-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  277nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127627(5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-...)
Affinity DataKi:  317nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127640(5-(2-Chloro-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  366nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127629(5-(4'-Iodo-biphenyl-4-ylmethylene)-3-aza-tricyclo[...)
Affinity DataKi:  377nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127643(5-(3',5'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  383nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127633(5-(2',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  393nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127636(5-(4'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  417nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  423nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127633(5-(2',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  466nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127627(5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-...)
Affinity DataKi:  531nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127628(5-(4-Pyrrol-1-yl-benzylidene)-3-aza-tricyclo[4.4.2...)
Affinity DataKi:  568nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127629(5-(4'-Iodo-biphenyl-4-ylmethylene)-3-aza-tricyclo[...)
Affinity DataKi:  660nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127624(5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-t...)
Affinity DataKi:  674nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127636(5-(4'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  739nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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