Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50013611
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132483(CHEMBL108043 | Pentyl-(1-phenethyloxy-4,5-dihydro-...)
Affinity DataKi:  4.90E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor was measured through displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132481((1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl)-pentyl-...)
Affinity DataKi:  5.50E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor was measured through displacement of [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50132483(CHEMBL108043 | Pentyl-(1-phenethyloxy-4,5-dihydro-...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor was measured through displacement of [3H]-RX-821002More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50132481((1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl)-pentyl-...)
Affinity DataKi:  3.00E+4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor was measured through displacement of [3H]-RX-821002More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132483(CHEMBL108043 | Pentyl-(1-phenethyloxy-4,5-dihydro-...)
Affinity DataIC50: <100nMAssay Description:Inhibitory activity against N-methyl-D-aspartate glutamate receptor 2A in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132481((1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl)-pentyl-...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against N-methyl-D-aspartate glutamate receptor 2A in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132483(CHEMBL108043 | Pentyl-(1-phenethyloxy-4,5-dihydro-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory activity against N-methyl-D-aspartate glutamate receptor 2B in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50132481((1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl)-pentyl-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against N-methyl-D-aspartate glutamate receptor 2B in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed