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Found 21 Enz. Inhib. hit(s) with all data for entry = 50036009
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000784(2-(3,4-Dichloro-phenyl)-N-methyl-N-(7-pyrrolidin-1...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  15nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000785(2-(3,4-Dichloro-phenyl)-N-methyl-N-(5-oxo-2-pyrrol...)
Affinity DataKi:  78nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000782(2-(3,4-Dichloro-phenyl)-N-methyl-N-(8-pyrrolidin-1...)
Affinity DataKi:  94nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000786(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  109nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  252nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000784(2-(3,4-Dichloro-phenyl)-N-methyl-N-(7-pyrrolidin-1...)
Affinity DataKi:  702nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  825nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000781(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000784(2-(3,4-Dichloro-phenyl)-N-methyl-N-(7-pyrrolidin-1...)
Affinity DataKi:  1.64E+3nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000781(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  2.61E+3nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000786(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  3.15E+3nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000782(2-(3,4-Dichloro-phenyl)-N-methyl-N-(8-pyrrolidin-1...)
Affinity DataKi:  5.21E+3nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  9.40E+3nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000786(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  9.51E+3nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000781(2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-...)
Affinity DataKi:  1.23E+4nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000785(2-(3,4-Dichloro-phenyl)-N-methyl-N-(5-oxo-2-pyrrol...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity against opioid receptor mu from guinea pig brain membranes using [3H]naloxone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000782(2-(3,4-Dichloro-phenyl)-N-methyl-N-(8-pyrrolidin-1...)
Affinity DataKi:  1.75E+4nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000785(2-(3,4-Dichloro-phenyl)-N-methyl-N-(5-oxo-2-pyrrol...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed