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Found 21 Enz. Inhib. hit(s) with all data for entry = 50036004
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002099(CHEMBL366965 | Dimethyl-[3-(2-methyl-6H-dibenzo[b,...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002087(4-(1-Methyl-piperidin-4-ylidene)-4,9-dihydro-1-thi...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002083(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002102(2-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  0.630nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002103(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002095(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002085(CHEMBL304185 | [11-(4-Dimethylamino-butylidene)-6,...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002086(11-(3-Pyrrolidin-1-yl-propylidene)-6,11-dihydro-di...)
Affinity DataKi:  5nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002093(CHEMBL65699 | [11-(3-Dimethylamino-propylidene)-6,...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002097(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  5.80nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002098(11-(4-Dimethylamino-butylidene)-6,11-dihydro-diben...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002092(11-(3-Thiomorpholin-4-yl-propylidene)-6,11-dihydro...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002100(11-(3-Diethylamino-propylidene)-6,11-dihydro-diben...)
Affinity DataKi:  10nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002088(CHEMBL302005 | [11-(2-Dimethylamino-ethylidene)-6,...)
Affinity DataKi:  11nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002101(11-(2-Dimethylamino-ethylidene)-6,11-dihydro-diben...)
Affinity DataKi:  12nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002084(11-(2-Dimethylamino-ethylsulfanyl)-6,11-dihydro-di...)
Affinity DataKi:  14nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002089(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  15nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002096(ALO-4943A | CHEMBL1719 | KW-4679 | OLOPATADINE HYD...)
Affinity DataKi:  16nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002091(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  20nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002090(11-(3-Dimethylamino-propylidene)-6,11-dihydro-dibe...)
Affinity DataKi:  24nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002094(3-[11-(3-Dimethylamino-propylidene)-6,11-dihydro-d...)
Affinity DataKi:  29nMAssay Description:Binding affinity for histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand at 0.1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed