Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50000160
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002186(CHEMBL440987 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  0.00420nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002182(CHEMBL415617 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  0.00670nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002185(CHEMBL438741 | Tyr-Gly-Gly-Phe-Leu-Lys(Ac)-Arg-Ile...)
Affinity DataKi:  0.0180nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002181(CHEMBL266717 | Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Ile-Arg...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002183(CHEMBL266515 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile-Arg...)
Affinity DataKi:  0.0210nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002185(CHEMBL438741 | Tyr-Gly-Gly-Phe-Leu-Lys(Ac)-Arg-Ile...)
Affinity DataKi:  0.0240nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002178(CHEMBL440446 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002186(CHEMBL440987 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  0.0430nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002182(CHEMBL415617 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  0.0460nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002178(CHEMBL440446 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  0.0530nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002183(CHEMBL266515 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile-Arg...)
Affinity DataKi:  0.0550nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002179(CHEMBL263597 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002181(CHEMBL266717 | Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Ile-Arg...)
Affinity DataKi:  0.0750nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002180(CHEMBL263583 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys(Ac)-Ile...)
Affinity DataKi:  0.140nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002179(CHEMBL263597 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of [3H]- bremazocine to opioid receptor kappa of guinea pig cerebral membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002180(CHEMBL263583 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys(Ac)-Ile...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002185(CHEMBL438741 | Tyr-Gly-Gly-Phe-Leu-Lys(Ac)-Arg-Ile...)
Affinity DataKi:  0.420nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002178(CHEMBL440446 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002180(CHEMBL263583 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys(Ac)-Ile...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002186(CHEMBL440987 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002183(CHEMBL266515 | Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile-Arg...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002182(CHEMBL415617 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Lys...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002179(CHEMBL263597 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002181(CHEMBL266717 | Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Ile-Arg...)
Affinity DataKi:  5.90nMAssay Description:Inhibition of [3H]-DPDPE to opioid receptor delta of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed