Compile Data Set for Download or QSAR
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Found 55 Enz. Inhib. hit(s) with all data for entry = 50000233
LigandPNGBDBM50230088(CHEMBL125786)
Affinity DataIC50:  58nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003292(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  90nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230079(CHEMBL126594)
Affinity DataIC50:  120nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230114(CHEMBL339961)
Affinity DataIC50:  150nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230103(CHEMBL126356)
Affinity DataIC50:  250nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230105(CHEMBL339446)
Affinity DataIC50:  300nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003285(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003265(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  330nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230098(CHEMBL127005)
Affinity DataIC50:  360nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003264(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  400nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003266((E)-3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-y...)
Affinity DataIC50:  440nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230115(CHEMBL338478)
Affinity DataIC50:  470nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003288(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  700nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003271(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  730nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230096(CHEMBL338517)
Affinity DataIC50:  810nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230085(CHEMBL126359)
Affinity DataIC50:  810nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230080(CHEMBL339860)
Affinity DataIC50:  820nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230109(CHEMBL127379)
Affinity DataIC50:  860nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230089(CHEMBL436594)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230083(CHEMBL444069)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003269(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003301((Z-isomer)-2-Benzyl-3-[2-butyl-3-(2-chloro-benzyl)...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230094(CHEMBL127308)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003282(2-(4-Amino-benzyl)-3-[2-butyl-3-(2-chloro-benzyl)-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230111(CHEMBL126501)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230087(CHEMBL339623)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003279(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230107(CHEMBL338067)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230116(CHEMBL338249)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230095(CHEMBL405525)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230108(CHEMBL126500)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230112(CHEMBL338690)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003254(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  1.00E+4nMAssay Description:Compound was evaluated for the inhibition of [125I]-AII specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230118(CHEMBL340917)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003290(CHEMBL39345 | [2-Butyl-3-(2-chloro-benzyl)-3H-imid...)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was evaluated for the inhibition of Angiotensin II receptor induced vasoconstriction of the rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230090(CHEMBL127916)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230086(CHEMBL339939)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230104(CHEMBL127515)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230102(CHEMBL127566)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230106(CHEMBL125341)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230101(CHEMBL127137)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230097(CHEMBL434254)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230113(CHEMBL435804)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230099(CHEMBL340433)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230084(CHEMBL338423)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230117(CHEMBL126357)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003278(3-[2-Butyl-3-(2-chloro-benzyl)-3H-imidazol-4-yl]-2...)
Affinity DataIC50:  2.56E+4nMAssay Description:Inhibition of [125I]-Angiotensin II receptor specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230091(CHEMBL340316)
Affinity DataIC50:  2.84E+4nMAssay Description:Compound was tested in vitro for binding affinity against human carbonic anhydrase II; (ki*10e-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230082(CHEMBL339121)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibition of [125I]angiotensin II specific binding to rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230110(CHEMBL353234)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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