Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50000265
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKi:  10nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKi:  80nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKi:  120nMAssay Description:Compound was tested for its binding affinity against the enzyme Tissue plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003740((Lactone IIa)N-[4-(2-Methylene-6-oxo-tetrahydro-py...)
Affinity DataKi:  120nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKi:  170nMAssay Description:Compound was tested for its binding affinity against the enzyme alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003742((Lactone1)N-[4-(6-Methylene-2-oxo-tetrahydro-pyran...)
Affinity DataKi:  350nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003739((Lactone3)N-[4-(4-Guanidino-phenyl)-6-methylene-2-...)
Affinity DataKi:  460nMAssay Description:Compound was tested for its binding affinity against the enzyme alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKi:  670nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKi:  670nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKi:  1.19E+3nMAssay Description:Compound was tested for its binding affinity against the enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003741(CHEMBL137269 | N-[4-(2-Iodomethylene-6-oxo-tetrahy...)
Affinity DataKi:  4.28E+3nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003739((Lactone3)N-[4-(4-Guanidino-phenyl)-6-methylene-2-...)
Affinity DataKi:  6.00E+3nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003741(CHEMBL137269 | N-[4-(2-Iodomethylene-6-oxo-tetrahy...)
Affinity DataKi:  7.83E+3nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003740((Lactone IIa)N-[4-(2-Methylene-6-oxo-tetrahydro-py...)
Affinity DataKi:  9.40E+3nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003739((Lactone3)N-[4-(4-Guanidino-phenyl)-6-methylene-2-...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKi:  1.48E+4nMAssay Description:Compound was tested for its binding affinity against the enzyme thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKi:  1.87E+4nMAssay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003742((Lactone1)N-[4-(6-Methylene-2-oxo-tetrahydro-pyran...)
Affinity DataKi:  3.79E+4nMAssay Description:Compound was tested for its binding affinity against the enzyme thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003742((Lactone1)N-[4-(6-Methylene-2-oxo-tetrahydro-pyran...)
Affinity DataKi:  4.66E+5nMAssay Description:Compound was tested for its binding affinity against the enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003739((Lactone3)N-[4-(4-Guanidino-phenyl)-6-methylene-2-...)
Affinity DataKon:  0.000250M-1s-1Assay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003741(CHEMBL137269 | N-[4-(2-Iodomethylene-6-oxo-tetrahy...)
Affinity DataKon:  0.000330M-1s-1Assay Description:Compound was tested for its binding affinity against the enzyme trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003739((Lactone3)N-[4-(4-Guanidino-phenyl)-6-methylene-2-...)
Affinity DataKon:  0.0000330M-1s-1Assay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003740((Lactone IIa)N-[4-(2-Methylene-6-oxo-tetrahydro-py...)
Affinity DataKon:  0.0000330M-1s-1Assay Description:Compound was tested for its binding affinity against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003742((Lactone1)N-[4-(6-Methylene-2-oxo-tetrahydro-pyran...)
Affinity DataKon:  0.000730M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003738((lactone 2)N-[4-(6-Iodomethylene-2-oxo-tetrahydro-...)
Affinity DataKon:  0.000220M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003742((Lactone1)N-[4-(6-Methylene-2-oxo-tetrahydro-pyran...)
Affinity DataKon:  0.000100M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKon:  0.0000130M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003737((Lactone4)N-[4-(4-Guanidino-phenyl)-6-iodomethylen...)
Affinity DataKon:  0.0000830M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against the enzyme Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50003740((Lactone IIa)N-[4-(2-Methylene-6-oxo-tetrahydro-py...)
Affinity DataKon:  0.000150M-1s-1Assay Description:Compound was tested for the rate constant of deacylation against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed