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Found 23 Enz. Inhib. hit(s) with all data for entry = 50042230
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM81471(CAS_91-81-6 | NSC_5587 | Tripelennamine)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataIC50:  158nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422502(CHEMBL158352)
Affinity DataIC50:  251nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422503(CHEMBL157217)
Affinity DataIC50:  398nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422500(CHEMBL157273)
Affinity DataIC50:  398nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50407521(CHEMBL94249)
Affinity DataIC50:  501nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422494(CHEMBL152126)
Affinity DataIC50:  631nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22864(2-[2-(3,3-diphenylpropyl)-1H-imidazol-4-yl]ethan-1...)
Affinity DataIC50:  794nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422495(CHEMBL155188)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50403672(CHEMBL24665)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22865(2-(2-aminoethyl)pyridine | 2-(pyridin-2-yl)ethan-1...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422497(CHEMBL152122)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422496(CHEMBL156071)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422501(CHEMBL345185)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422504(CHEMBL155314)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM86172(2-(3-Chlorophenyl)histamine)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422506(CHEMBL157842)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422493(CHEMBL359122)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50407520(CHEMBL90063)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422499(CHEMBL152221)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422498(CHEMBL154566)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422505(CHEMBL154068)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed