Compile Data Set for Download or QSAR
maximum 50k data
Found 70 Enz. Inhib. hit(s) with all data for entry = 50014034
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137438(5-Methanesulfonyl-2-[5-(4-methoxy-phenyl)-3-triflu...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137423(2-(4-Chloro-3-difluoromethyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137420(2-[5-(4-Ethoxy-phenyl)-3-trifluoromethyl-pyrazol-1...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137442(2-[3-Difluoromethyl-5-(3-fluoro-4-methoxy-phenyl)-...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137435(2-(4-Chloro-5-phenyl-3-trifluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137439(2-[5-(2-Fluoro-4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137424(2-[4-Chloro-5-(3-chloro-4-methoxy-phenyl)-3-difluo...)
Affinity DataIC50:  62nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137411(2-[3-Difluoromethyl-5-(4-methoxy-phenyl)-pyrazol-1...)
Affinity DataIC50:  64nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137437(5-Methanesulfonyl-2-[5-(4-methylsulfanyl-phenyl)-3...)
Affinity DataIC50:  69nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137427(2-(4-Bromo-3-difluoromethyl-5-phenyl-pyrazol-1-yl)...)
Affinity DataIC50:  80nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137440(CHEMBL176934 | {4-[2-(5-Methanesulfonyl-pyridin-2-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137428(2-[3-Difluoromethyl-5-(4-methylsulfanyl-phenyl)-py...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137414(2-[5-(4-Chloro-phenyl)-3-difluoromethyl-pyrazol-1-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137420(2-[5-(4-Ethoxy-phenyl)-3-trifluoromethyl-pyrazol-1...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137412(5-Methanesulfonyl-2-(4-methyl-5-phenyl-3-trifluoro...)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137434(2-[3-Difluoromethyl-5-(4-methoxy-3-methyl-phenyl)-...)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137418(2-(3-Difluoromethyl-5-p-tolyl-pyrazol-1-yl)-5-meth...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137432(2-(3-Difluoromethyl-4-methyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137411(2-[3-Difluoromethyl-5-(4-methoxy-phenyl)-pyrazol-1...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137416(2-(5-(4-fluorophenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137413(2-[5-(4-Chloro-phenyl)-3-trifluoromethyl-pyrazol-1...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137415(5-Methanesulfonyl-2-[5-(4-methoxy-3-methyl-phenyl)...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137410(2-[5-(4-Bromo-phenyl)-3-difluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137441(2-[5-(3-Chloro-4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137429(2-[3-Difluoromethyl-5-(4-fluoro-phenyl)-pyrazol-1-...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137425(2-(3-(difluoromethyl)-5-phenyl-1H-pyrazol-1-yl)-5-...)
Affinity DataIC50:  310nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137421(2-[5-(3-Fluoro-4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  310nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137436(2-[5-(3-Chloro-4-methoxy-phenyl)-3-difluoromethyl-...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137423(2-(4-Chloro-3-difluoromethyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137422(2-[3-Difluoromethyl-5-(2-fluoro-4-methoxy-phenyl)-...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137417(2-[3-Difluoromethyl-5-(4-ethyl-phenyl)-pyrazol-1-y...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137433(5-(methylsulfonyl)-2-(5-phenyl-3-(trifluoromethyl)...)
Affinity DataIC50:  410nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137419(2-[5-(4-Bromo-phenyl)-3-trifluoromethyl-pyrazol-1-...)
Affinity DataIC50:  450nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50057583(4-[3-Difluoromethyl-5-(3-fluoro-4-methoxy-phenyl)-...)
Affinity DataIC50:  630nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137438(5-Methanesulfonyl-2-[5-(4-methoxy-phenyl)-3-triflu...)
Affinity DataIC50:  830nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137428(2-[3-Difluoromethyl-5-(4-methylsulfanyl-phenyl)-py...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137410(2-[5-(4-Bromo-phenyl)-3-difluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137424(2-[4-Chloro-5-(3-chloro-4-methoxy-phenyl)-3-difluo...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137431(2-[5-(3-Bromo-4-methoxy-phenyl)-3-trifluoromethyl-...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137437(5-Methanesulfonyl-2-[5-(4-methylsulfanyl-phenyl)-3...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137430(2-[3-Difluoromethyl-5-(4-propyl-phenyl)-pyrazol-1-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137427(2-(4-Bromo-3-difluoromethyl-5-phenyl-pyrazol-1-yl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137439(2-[5-(2-Fluoro-4-methoxy-phenyl)-3-trifluoromethyl...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  5.57E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137435(2-(4-Chloro-5-phenyl-3-trifluoromethyl-pyrazol-1-y...)
Affinity DataIC50:  7.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137426(2-[3-Difluoromethyl-5-(4-isopropyl-phenyl)-pyrazol...)
Affinity DataIC50:  8.10E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137432(2-(3-Difluoromethyl-4-methyl-5-phenyl-pyrazol-1-yl...)
Affinity DataIC50:  9.10E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137442(2-[3-Difluoromethyl-5-(3-fluoro-4-methoxy-phenyl)-...)
Affinity DataIC50:  9.90E+3nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137418(2-(3-Difluoromethyl-5-p-tolyl-pyrazol-1-yl)-5-meth...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibitory activity against cannine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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