Compile Data Set for Download or QSAR
maximum 50k data
Found 154 Enz. Inhib. hit(s) with all data for entry = 50014049
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137582(CHEMBL292930 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137587(3-[1-(3-Morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137576(3-[1-{3-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-4,5,...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137573(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137574(3-[1-{3-[3-(4-Methyl-piperazin-1-yl)-propyl]-4,5,6...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137578(CHEMBL300853 | [4-(3-{2-[5-Ethanesulfonyl-2-oxo-1,...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137571(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137583(3-[1-(3-{3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-pr...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137570(CHEMBL291759 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137582(CHEMBL292930 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137584(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137581(5-Ethanesulfonyl-3-[1-{3-[3-(4-hydroxy-piperidin-1...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137569(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137573(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137583(3-[1-(3-{3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-pr...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137580(3-[1-[3-(3-Morpholin-4-yl-propyl)-4,5,6,7-tetrahyd...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137572(5-Ethanesulfonyl-3-[1-{3-[3-(4-methyl-piperazin-1-...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137587(3-[1-(3-Morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137569(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137591(5-Ethanesulfonyl-3-[1-(3-{3-[4-(2-hydroxy-ethyl)-p...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137573(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against Fyn tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137576(3-[1-{3-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-4,5,...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137584(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137580(3-[1-[3-(3-Morpholin-4-yl-propyl)-4,5,6,7-tetrahyd...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137587(3-[1-(3-Morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against Vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137571(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against Fyn tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137574(3-[1-{3-[3-(4-Methyl-piperazin-1-yl)-propyl]-4,5,6...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137570(CHEMBL291759 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137585(5-Ethanesulfonyl-3-[1-(3-morpholin-4-ylmethyl-4,5,...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137581(5-Ethanesulfonyl-3-[1-{3-[3-(4-hydroxy-piperidin-1...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137573(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137578(CHEMBL300853 | [4-(3-{2-[5-Ethanesulfonyl-2-oxo-1,...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137591(5-Ethanesulfonyl-3-[1-(3-{3-[4-(2-hydroxy-ethyl)-p...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137587(3-[1-(3-Morpholin-4-ylmethyl-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against Lck tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137569(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137570(CHEMBL291759 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137571(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137580(3-[1-[3-(3-Morpholin-4-yl-propyl)-4,5,6,7-tetrahyd...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137573(3-{2-[5-Methylsulfamoyl-2-oxo-1,2-dihydro-indol-(3...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Lck tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137574(3-[1-{3-[3-(4-Methyl-piperazin-1-yl)-propyl]-4,5,6...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137571(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137583(3-[1-(3-{3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-pr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Fyn tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137585(5-Ethanesulfonyl-3-[1-(3-morpholin-4-ylmethyl-4,5,...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137582(CHEMBL292930 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Lck tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137613(5-Ethanesulfonyl-3-[1-[3-(3-morpholin-4-yl-propyl)...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137585(5-Ethanesulfonyl-3-[1-(3-morpholin-4-ylmethyl-4,5,...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against Yes tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137584(3-[1-[3-(3-Dimethylamino-propyl)-4,5,6,7-tetrahydr...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against Lck tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137582(CHEMBL292930 | [4-(3-{2-[5-Methylsulfamoyl-2-oxo-1...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137572(5-Ethanesulfonyl-3-[1-{3-[3-(4-methyl-piperazin-1-...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against cellular Src protein tryrosine kinase using the actin ring assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Sugen

Curated by ChEMBL
LigandPNGBDBM50137569(3-{2-[5-Ethanesulfonyl-2-oxo-1,2-dihydro-indol-(3Z...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against Fyn tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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